Compile Data Set for Download or QSAR
Report error Found 86 Enz. Inhib. hit(s) with all data for entry = 50021127
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221380(N-(4-{4-[benzyl(phenyl)amino]piperidin-1-yl}butyln...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50119380(CHEMBL540612 | N-(4-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221374(N-(4-{4-[(4-chlorophenyl)phenylmethyl]piperazin-1-...)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221376(benzo[b]thiophene-2-carboxylic acid {4-[4-(8-chlor...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221369(N-(4-{4-[(4-chlorophenyl)phenylmethyl]piperazin-1-...)
Affinity DataKi:  2.82nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221400(N-(4-(4-((2-methoxyphenyl)(phenyl)methyl)piperazin...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221367(naphthalene-2-carboxylic acid {4-[4-(8-chloro-5,6-...)
Affinity DataKi:  6.01nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221387(N-[4-(4-diphenylmethylpiperazin-1-yl)butyl]cinnami...)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221366(N-(4-(3,4-dihydroisoquinolin-2(1H)-yl)butyl)cinnam...)
Affinity DataKi:  8.72nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221360(N-(4-(4-(2-methoxyphenylamino)piperidin-1-yl)butyl...)
Affinity DataKi:  10.8nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221391(naphthalene-2-carboxylic acid {4-[4-(10-oxo-9,10-d...)
Affinity DataKi:  10.9nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221381(N-{4-[4-(diphenylmethyl)piperazin-1-yl]butyl}napht...)
Affinity DataKi:  11.1nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221365(N-(4-{4-[(4-chlorophenyl)phenylmethyl]piperazin-1-...)
Affinity DataKi:  12.3nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221368(N-(4-(4-(bis(2-methoxyphenyl)methyl)piperazin-1-yl...)
Affinity DataKi:  15.2nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221394(N-(4-(4-(bis(2-methoxyphenyl)methyl)piperazin-1-yl...)
Affinity DataKi:  15.2nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221361(N-(4-{4-[(4-chlorophenyl)phenylmethyl)piperazin-1-...)
Affinity DataKi:  17.7nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221384(N-(4-(4-(2-methoxyphenylamino)piperidin-1-yl)butyl...)
Affinity DataKi:  18.4nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221399(N-(4-(4-(bis(2-methoxyphenyl)methyl)piperazin-1-yl...)
Affinity DataKi:  22.8nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221393(N-(4-{4-[(4-chlorophenyl)phenylmethyl]piperazin-1-...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221386(N-[4-(4-diphenylmethylpiperazin-1-yl)butyl]thiophe...)
Affinity DataKi:  28.4nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221377(N-[4-(4-diphenylmethylpiperazin-1-yl)butyl]cyclohe...)
Affinity DataKi:  30.2nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221359(N-[4-(4-diphenylmethylpiperazin-1-yl)butyl]benzo-[...)
Affinity DataKi:  30.3nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221395(N-(4-{4-[benzyl(phenyl)amino]piperidin-1-yl}butyl)...)
Affinity DataKi:  31.1nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221382(N-{4-[4-(diphenylmethyl)-1,4-diazepan-1-yl]butyl}-...)
Affinity DataKi:  32.6nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221389(N-{4-[4-(diphenylmethyl)-1,4-diazepan-1-yl]butyl}-...)
Affinity DataKi:  36.9nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221371(N-(4-{4-[(4-chlorophenyl)phenylmethyl]piperazin-1-...)
Affinity DataKi:  38.9nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221385(N-{4-[4-(diphenylmethyl)-1,4-diazepan-1-yl]butyl}-...)
Affinity DataKi:  40.9nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221396(N-(4-{4-[(4-chlorophenyl)phenylmethyl]-1,4-diazepa...)
Affinity DataKi:  42.9nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221375(N-{4-[4-(diphenylmethyl)piperazin-1-yl]butyl}isoin...)
Affinity DataKi:  47.3nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221363(N-[4-(2,3,4,5,10,15-hexahydro-1H-dibenzo[b:e]-pyra...)
Affinity DataKi:  50.2nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50119380(CHEMBL540612 | N-(4-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221388(N-{4-[4-(10-oxo-9,10-dihydro-4H-benzo[4,5]cyclohep...)
Affinity DataKi:  99.1nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221362(N-{4-[4-(N'-benzyl-N0-phenylamino)piperidin-1-yl]b...)
Affinity DataKi:  128nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221370(N-{4-[4-(diphenylmethyl)-1,4-diazepan-1-yl]butyl}i...)
Affinity DataKi:  133nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221382(N-{4-[4-(diphenylmethyl)-1,4-diazepan-1-yl]butyl}-...)
Affinity DataKi:  136nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221371(N-(4-{4-[(4-chlorophenyl)phenylmethyl]piperazin-1-...)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221385(N-{4-[4-(diphenylmethyl)-1,4-diazepan-1-yl]butyl}-...)
Affinity DataKi:  161nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221384(N-(4-(4-(2-methoxyphenylamino)piperidin-1-yl)butyl...)
Affinity DataKi:  163nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221365(N-(4-{4-[(4-chlorophenyl)phenylmethyl]piperazin-1-...)
Affinity DataKi:  189nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221396(N-(4-{4-[(4-chlorophenyl)phenylmethyl]-1,4-diazepa...)
Affinity DataKi:  226nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221367(naphthalene-2-carboxylic acid {4-[4-(8-chloro-5,6-...)
Affinity DataKi:  252nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221392(N-[4-(2,3,4,5,10,15-hexahydro-1H-dibenzo[b:e]-pyra...)
Affinity DataKi:  258nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221394(N-(4-(4-(bis(2-methoxyphenyl)methyl)piperazin-1-yl...)
Affinity DataKi:  313nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221378(N-{4-[4-(diphenylmethyl)-1,4-diazepan-1-yl]butyl}-...)
Affinity DataKi:  340nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221363(N-[4-(2,3,4,5,10,15-hexahydro-1H-dibenzo[b:e]-pyra...)
Affinity DataKi:  429nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221377(N-[4-(4-diphenylmethylpiperazin-1-yl)butyl]cyclohe...)
Affinity DataKi:  435nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221381(N-{4-[4-(diphenylmethyl)piperazin-1-yl]butyl}napht...)
Affinity DataKi:  457nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221364(N-[4-(2,3,4,5,10,15-hexahydro-1H-dibenzo[b:e]-pyra...)
Affinity DataKi:  497nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221390(N-[4-(2,3,4,5,10,15-hexahydro-1H-dibenzo[b: e]pyra...)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50221364(N-[4-(2,3,4,5,10,15-hexahydro-1H-dibenzo[b:e]-pyra...)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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