Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50021171
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataIC50:  2.32E+3nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM50221762(6-hydroxy-2-phenyl-4H-pyrido[1,2-a]pyrimidin-4-one...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM50221751(2-(3,4-dihydroxyphenyl)-6-hydroxy-4H-pyrido[1,2-a]...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM50221748(2-(3,4-dimethoxyphenyl)-6-hydroxy-4H-pyrido[1,2-a]...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM50221752(6-hydroxy-2-(4-hydroxyphenyl)-4H-pyrido[1,2-a]pyri...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM50221756(2-(3,4-dimethoxyphenyl)-4H-pyrido[1,2-a]pyrimidin-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM50221757(2-(3,4-dihydroxyphenyl)-9-hydroxy-4H-pyrido[1,2-a]...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM50221758(2-benzyl-6-hydroxy-4H-pyrido[1,2-a]pyrimidin-4-one...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM50221759(2-(4-hydroxybenzyl)-6-hydroxy-4H-pyrido[1,2-a]pyri...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM50221754(2-(4-methoxybenzyl)-6-hydroxy-4H-pyrido[1,2-a]pyri...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM50221753(2-phenyl-4H-pyrido[1,2-a]pyrimidin-4-one | CHEMBL2...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM50221760(2-(4-methoxyphenyl)-4H-pyrido[1,2-a]pyrimidin-4-on...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM50221755(2-(4-hydroxyphenyl)-4H-pyrido[1,2-a]pyrimidin-4-on...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM50221763(9-hydroxy-2-(4-hydroxyphenyl)-4H-pyrido[1,2-a]pyri...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM50221765(2-(3,4-dimethoxybenzyl)-6-hydroxy-4H-pyrido[1,2-a]...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM50221747(6-hydroxy-2-(4-methoxyphenyl)-4H-pyrido[1,2-a]pyri...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM50221764(2-(3,4-dimethoxyphenyl)-9-hydroxy-4H-pyrido[1,2-a]...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM50221766(9-hydroxy-2-phenyl-4H-pyrido[1,2-a]pyrimidin-4-one...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM50221761(9-hydroxy-2-(4-methoxyphenyl)-4H-pyrido[1,2-a]pyri...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM50221749(2-(3,4-dihydroxyphenyl)-4H-pyrido[1,2-a]pyrimidin-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM50221750(2-(3,4-dihydroxybenzyl)-6-hydroxy-4H-pyrido[1,2-a]...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ALR1 in Sprague-Dawley Albino rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed