Compile Data Set for Download or QSAR
maximum 50k data
Found 51 Enz. Inhib. hit(s) with all data for entry = 50021242
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM25036(CHEMBL393525 | N'-[(1E)-{6-bromoimidazo[1,2-a]pyri...)
Affinity DataIC50:  7.80nMAssay Description:Inhibition of human recombinant p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM25036(CHEMBL393525 | N'-[(1E)-{6-bromoimidazo[1,2-a]pyri...)
Affinity DataIC50:  340nMAssay Description:Inhibition of human recombinant p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222534(CHEMBL240335 | N'-(isoquinolin-4-ylmethylene)-N,2-...)
Affinity DataIC50:  800nMAssay Description:Inhibition of human recombinant p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222539(CHEMBL239050 | N'-(imidazo[1,2-a]pyridin-3-ylmethy...)
Affinity DataIC50:  860nMAssay Description:Inhibition of human recombinant p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM25036(CHEMBL393525 | N'-[(1E)-{6-bromoimidazo[1,2-a]pyri...)
Affinity DataIC50:  910nMAssay Description:Inhibition of human recombinant p110deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222538(CHEMBL240336 | N'-((6-bromoisoquinolin-4-yl)methyl...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human recombinant p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222527(CHEMBL393747 | N,2-dimethyl-5-nitro-N'-(quinolin-4...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of human recombinant p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222534(CHEMBL240335 | N'-(isoquinolin-4-ylmethylene)-N,2-...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of human recombinant p110deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222529(CHEMBL392070 | N'-(benzo[c]isoxazol-3-ylmethylene)...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human recombinant p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222539(CHEMBL239050 | N'-(imidazo[1,2-a]pyridin-3-ylmethy...)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of human recombinant p110deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222538(CHEMBL240336 | N'-((6-bromoisoquinolin-4-yl)methyl...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of human recombinant p110deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222535(CHEMBL413803 | N,2-dimethyl-N'-(naphthalen-1-ylmet...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222536(CHEMBL397105 | N'-((7-bromoisoquinolin-4-yl)methyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222537(CHEMBL240118 | N,2-dimethyl-5-nitro-N'-(quinolin-3...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222532(CHEMBL239475 | N,2-dimethyl-N'-((1-methyl-1H-indol...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222535(CHEMBL413803 | N,2-dimethyl-N'-(naphthalen-1-ylmet...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222529(CHEMBL392070 | N'-(benzo[c]isoxazol-3-ylmethylene)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222536(CHEMBL397105 | N'-((7-bromoisoquinolin-4-yl)methyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222533(CHEMBL397796 | N,2-dimethyl-N'-((1-methyl-1H-imida...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222537(CHEMBL240118 | N,2-dimethyl-5-nitro-N'-(quinolin-3...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222528(CHEMBL239052 | N'-(imidazo[1,5-a]pyridin-1-ylmethy...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222538(CHEMBL240336 | N'-((6-bromoisoquinolin-4-yl)methyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222531(CHEMBL413802 | N'-(benzo[b]thiophen-3-ylmethylene)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222524(CHEMBL392071 | N'-(benzofuran-3-ylmethylene)-N,2-d...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222524(CHEMBL392071 | N'-(benzofuran-3-ylmethylene)-N,2-d...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222533(CHEMBL397796 | N,2-dimethyl-N'-((1-methyl-1H-imida...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222527(CHEMBL393747 | N,2-dimethyl-5-nitro-N'-(quinolin-4...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222525(CHEMBL239051 | N,2-dimethyl-5-nitro-N'-((5,6,7,8-t...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222527(CHEMBL393747 | N,2-dimethyl-5-nitro-N'-(quinolin-4...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222525(CHEMBL239051 | N,2-dimethyl-5-nitro-N'-((5,6,7,8-t...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222526(CHEMBL397780 | N'-((8-bromoisoquinolin-4-yl)methyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222539(CHEMBL239050 | N'-(imidazo[1,2-a]pyridin-3-ylmethy...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222531(CHEMBL413802 | N'-(benzo[b]thiophen-3-ylmethylene)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222530(CHEMBL393526 | N'-(imidazo[1,5-a]pyridin-3-ylmethy...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222525(CHEMBL239051 | N,2-dimethyl-5-nitro-N'-((5,6,7,8-t...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222526(CHEMBL397780 | N'-((8-bromoisoquinolin-4-yl)methyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222531(CHEMBL413802 | N'-(benzo[b]thiophen-3-ylmethylene)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222528(CHEMBL239052 | N'-(imidazo[1,5-a]pyridin-1-ylmethy...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222537(CHEMBL240118 | N,2-dimethyl-5-nitro-N'-(quinolin-3...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222535(CHEMBL413803 | N,2-dimethyl-N'-(naphthalen-1-ylmet...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222534(CHEMBL240335 | N'-(isoquinolin-4-ylmethylene)-N,2-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222532(CHEMBL239475 | N,2-dimethyl-N'-((1-methyl-1H-indol...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222533(CHEMBL397796 | N,2-dimethyl-N'-((1-methyl-1H-imida...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222532(CHEMBL239475 | N,2-dimethyl-N'-((1-methyl-1H-indol...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222530(CHEMBL393526 | N'-(imidazo[1,5-a]pyridin-3-ylmethy...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222529(CHEMBL392070 | N'-(benzo[c]isoxazol-3-ylmethylene)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222530(CHEMBL393526 | N'-(imidazo[1,5-a]pyridin-3-ylmethy...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222524(CHEMBL392071 | N'-(benzofuran-3-ylmethylene)-N,2-d...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222528(CHEMBL239052 | N'-(imidazo[1,5-a]pyridin-1-ylmethy...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50222536(CHEMBL397105 | N'-((7-bromoisoquinolin-4-yl)methyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant p110alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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