Compile Data Set for Download or QSAR
Report error Found 62 Enz. Inhib. hit(s) with all data for entry = 50021291
LigandPNGBDBM50222985(3,6-diethyl-N-((1R,2S)-2-(2-fluoroethoxy)-2,3-dihy...)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223023(5-(4,6-dimethylpyridin-2-yloxy)-N-((1R,2S)-2-ethox...)
Affinity DataKi:  22nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222980(3,6-diethyl-N-((1R,2S)-2-isopropoxy-2,3-dihydro-1H...)
Affinity DataKi:  22nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223004(3,6-diethyl-5-(4-methylpyridin-2-yloxy)-N-((1R,2S)...)
Affinity DataKi:  30nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223002(N-((1R,2S)-2-ethoxy-2,3-dihydro-1H-inden-1-yl)-3,6...)
Affinity DataKi:  35nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223033(3,6-diethyl-N-((1R,2S)-2-(2-fluoroethoxy)-2,3-dihy...)
Affinity DataKi:  51nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223020(N-((1R,2S)-2-ethoxy-2,3-dihydro-1H-inden-1-yl)-3,6...)
Affinity DataKi:  53nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223030(5-(4,6-dimethylpyridin-2-yloxy)-3,6-diethyl-N-((1R...)
Affinity DataKi:  58nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223015(3,6-diethyl-5-(4-methylpyridin-2-yloxy)-N-(1-pheny...)
Affinity DataKi:  59nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222977(N-((1R,2S)-2-(cyclopentyloxy)-2,3-dihydro-1H-inden...)
Affinity DataKi:  67nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223017(2-((1R,2S)-1-(3,6-diethyl-5-(4-methylpyridin-2-ylo...)
Affinity DataKi:  82nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223028(N2-(3,5-dichloropyridin-2-yl)-3,6-diethyl-N5-(pent...)
Affinity DataKi:  115nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222986(N-((1R,2S)-2-cyclopropoxy-2,3-dihydro-1H-inden-1-y...)
Affinity DataKi:  214nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222975(3,6-diethyl-N-((1R,2S)-2-methoxy-2,3-dihydro-1H-in...)
Affinity DataKi:  222nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222979(3,6-diethyl-5-(4-methylpyridin-2-yloxy)-N-(1-pheny...)
Affinity DataKi:  251nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222991(3,6-diethyl-N-((1R,2S)-2-(2-fluoroethoxy)-2,3-dihy...)
Affinity DataKi:  266nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222998(3,6-diethyl-N-(2-isopropoxy-1-phenylethyl)-5-(4-me...)
Affinity DataKi:  337nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223007(N-(2-ethoxy-1-phenylethyl)-3,6-diethyl-5-(4-methyl...)
Affinity DataKi:  384nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222978(3,6-dimethyl-5-(4-methylpyridin-2-yloxy)-N-(pentan...)
Affinity DataKi:  401nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223035(N-((1R,2S)-2-ethoxy-2,3-dihydro-1H-inden-1-yl)-3,6...)
Affinity DataKi:  436nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223032(N-((1R,2S)-2-ethoxy-2,3-dihydro-1H-inden-1-yl)-3,6...)
Affinity DataKi:  456nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223027(N-((1R,2S)-2-ethoxy-2,3-dihydro-1H-inden-1-yl)-3,6...)
Affinity DataKi:  472nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223010(N-((1R,2S)-2-ethoxy-2,3-dihydro-1H-inden-1-yl)-3,6...)
Affinity DataKi:  509nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223005(3,6-diethyl-N-(2-methyl-1-phenylpropyl)-5-(4-methy...)
Affinity DataKi:  530nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222982(3,6-diethyl-5-(4-methylpyridin-2-yloxy)-N,N-diprop...)
Affinity DataKi:  711nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223019(3,6-dimethyl-5-(4-methylpyridin-2-yloxy)-N,N-dipro...)
Affinity DataKi:  1.19E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223013(N-(cyclopropylmethyl)-3,6-dimethyl-5-(4-methylpyri...)
Affinity DataKi:  1.21E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223025(N2-(3,5-dichloropyridin-2-yl)-3,6-diethyl-N5-((1R,...)
Affinity DataKi:  1.21E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223014(N-((1R,2S)-2-ethoxy-2,3-dihydro-1H-inden-1-yl)-3,6...)
Affinity DataKi:  1.22E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223031(3,6-diethyl-N-((1R,2S)-2-methoxy-2,3-dihydro-1H-in...)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222988(3,6-diethyl-N2-(pentan-3-yl)-N5-(2,4,6-trichloroph...)
Affinity DataKi:  1.54E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222995(N2-(3,5-dichloropyridin-2-yl)-3,6-diethyl-N5-((1R,...)
Affinity DataKi:  1.73E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223016((1R,2S)-1-(3,6-diethyl-5-(4-methylpyridin-2-yloxy)...)
Affinity DataKi:  2.02E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223003(3,6-dimethyl-5-(4-methylpyridin-2-yloxy)-N-(1-phen...)
Affinity DataKi:  2.12E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222976(3,6-dimethyl-N-(2-methyl-1-phenylpropyl)-5-(4-meth...)
Affinity DataKi:  2.38E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223034(3,6-diethyl-5-(3-methylpyridin-2-yloxy)-N-(1-pheny...)
Affinity DataKi:  2.43E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223024(N2-(4-chlorophenyl)-3,6-diethyl-N5-(pentan-3-yl)py...)
Affinity DataKi:  2.70E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222994(3,6-diethyl-N2-(6-methylpyridin-2-yl)-N5-(pentan-3...)
Affinity DataKi:  3.38E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222989(N2-(3,5-dichloropyridin-2-yl)-3,6-dimethyl-N5-(pen...)
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222984(2-(3,6-diethyl-5-(4-methylpyridin-2-yloxy)pyrazin-...)
Affinity DataKi:  4.69E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222983(N-((1S,2S)-2-ethoxy-2,3-dihydro-1H-inden-1-yl)-3,6...)
Affinity DataKi:  5.47E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222999(N-((1R,2R)-2-ethoxy-2,3-dihydro-1H-inden-1-yl)-3,6...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223036(3,6-diethyl-5-(4-methylpyridin-2-yloxy)-N-(pentan-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223006(N-((1R,2S)-2-(3,6-dimethylpyrazin-2-yloxy)-2,3-dih...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223000(N2-(3,5-dichloropyridin-2-yl)-N2,3,6-triethyl-N5-(...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223001(N-((1R,2S)-2-isopropoxy-2,3-dihydro-1H-inden-1-yl)...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223008(3,6-diethyl-N2-(5-nitropyridin-2-yl)-N5-(pentan-3-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223009(3,6-diethyl-N2-(4-methylpyridin-2-yl)-N5-(pentan-3...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50223012(N2-(2,4-dichlorophenyl)-3,6-diethyl-N5-(pentan-3-y...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222981(N2-(3,5-dichloropyridin-2-yl)-3,6-diethyl-N5-(1-ph...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in IMR32 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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