Compile Data Set for Download or QSAR
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Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50021302
TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223090(3-(4-(3-chloro-4-fluorophenylamino)quinazolin-6-yl...)
Affinity DataIC50:  14nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)
Affinity DataIC50:  23nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
MMDB
PDB3D3D Structure (crystal)

TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50095259((6,7-Dimethoxy-quinazolin-4-yl)-(3-ethynyl-phenyl)...)
Affinity DataIC50:  29nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)
Affinity DataIC50:  39nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
MMDB
PDB3D3D Structure (crystal)

TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223084(CHEMBL251498 | N-(3-chloro-4-fluorophenyl)-6-(3-mo...)
Affinity DataIC50:  50nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223082(CHEMBL251700 | N-(3-chloro-4-fluorophenyl)-6-(3-(p...)
Affinity DataIC50:  89nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223095(4-(4-(3-chloro-4-fluorophenylamino)quinazolin-6-yl...)
Affinity DataIC50:  95nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223092(5-(4-(3-chloro-4-fluorophenylamino)quinazolin-6-yl...)
Affinity DataIC50:  114nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223085(CHEMBL249509 | N-(3-chloro-4-fluorophenyl)-6-ethyn...)
Affinity DataIC50:  127nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223093(4-(4-(3-chloro-4-fluorophenylamino)quinazolin-6-yl...)
Affinity DataIC50:  152nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223088(4-(4-(3-chloro-4-fluorophenylamino)quinazolin-6-yl...)
Affinity DataIC50:  186nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223086(4-(3-(6,7-dimethoxyquinazolin-4-ylamino)phenyl)-2-...)
Affinity DataIC50:  206nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223094(CHEMBL249511 | N-(3-chloro-4-fluorophenyl)-6-(2-ph...)
Affinity DataIC50:  331nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223091(4-(3-(6,7-dimethoxyquinazolin-4-ylamino)phenyl)but...)
Affinity DataIC50:  402nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223087(6,7-dimethoxy-N-(3-(2-phenylethynyl)phenyl)quinazo...)
Affinity DataIC50:  921nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223089(5-(3-(6,7-dimethoxyquinazolin-4-ylamino)phenyl)pen...)
Affinity DataIC50:  1.36E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223096(CHEMBL398963 | N-(3-chloro-4-fluorophenyl)-6-(2-(t...)
Affinity DataIC50:  1.64E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Development Center For Biotechnology

Curated by ChEMBL
LigandPNGBDBM50223083(3-(3-(6,7-dimethoxyquinazolin-4-ylamino)phenyl)pro...)
Affinity DataIC50:  1.64E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed