Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50021355
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223615BDBM50223615(3-bromo-5-cyclohexyl-N-(pyridin-3-ylmethyl)pyrazol...)
Affinity DataIC50: 27nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223602BDBM50223602(N-(2-(5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo...)
Affinity DataIC50: 34nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223587BDBM50223587(3-bromo-5-(2-chlorophenyl)-N-((pyridin-3-yloxy)met...)
Affinity DataIC50: 35nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223567BDBM50223567(US8580782, 8 | CHEMBL401303 | 3-bromo-5-(2-chlorop...)
Affinity DataIC50: 54nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223590BDBM50223590(3-bromo-5-(2-fluorophenyl)-N-((pyridin-3-yloxy)met...)
Affinity DataIC50: 130nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223583BDBM50223583(3-bromo-5-(piperidin-3-yl)-N-(pyridin-3-ylmethyl)p...)
Affinity DataIC50: 180nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223580BDBM50223580(3-bromo-5-(2-chlorophenyl)-N-methylpyrazolo[1,5-a]...)
Affinity DataIC50: 247nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223591BDBM50223591(3-bromo-5-(furan-2-yl)-N-(pyridin-3-ylmethyl)pyraz...)
Affinity DataIC50: 310nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223578BDBM50223578(3-bromo-5-(piperidin-4-yl)-N-(pyridin-3-ylmethyl)p...)
Affinity DataIC50: 410nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223594BDBM50223594(3-bromo-5-isopropyl-N-(pyridin-3-ylmethyl)pyrazolo...)
Affinity DataIC50: 420nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223593BDBM50223593(3-bromo-5-(2-chlorophenyl)-N-(4-(methylsulfonyl)ph...)
Affinity DataIC50: 450nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223581BDBM50223581(3-bromo-N-(pyridin-3-ylmethyl)-5-(thiophen-2-yl)py...)
Affinity DataIC50: 480nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223595BDBM50223595(1-(3-bromo-7-(pyridin-3-ylmethylamino)pyrazolo[1,5...)
Affinity DataIC50: 500nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223586BDBM50223586(3-bromo-5-phenyl-N-(pyridin-3-ylmethyl)pyrazolo[1,...)
Affinity DataIC50: 570nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223609BDBM50223609(3-bromo-5-phenyl-N-((pyridin-3-yloxy)methyl)pyrazo...)
Affinity DataIC50: 600nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223568BDBM50223568(ethyl 3-bromo-7-(pyridin-3-ylmethylamino)pyrazolo[...)
Affinity DataIC50: 790nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223608BDBM50223608(3-bromo-5-ethyl-N-(pyridin-3-ylmethyl)pyrazolo[1,5...)
Affinity DataIC50: 920nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223605BDBM50223605(2-(5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223573BDBM50223573(3-bromo-5-cyclopropyl-N-(pyridin-3-ylmethyl)pyrazo...)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223577BDBM50223577(3-bromo-5-(methylthio)-N-(pyridin-3-ylmethyl)pyraz...)
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223601BDBM50223601(3-bromo-5-methoxy-N-(pyridin-3-ylmethyl)pyrazolo[1...)
Affinity DataIC50: 1.41E+3nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223592BDBM50223592(3-(methylthio)-5-phenyl-N-(pyridin-3-ylmethyl)pyra...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223607BDBM50223607(3-ethyl-5-phenyl-N-(pyridin-3-ylmethyl)pyrazolo[1,...)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223599BDBM50223599(3-bromo-5-methyl-N-(pyridin-3-ylmethyl)pyrazolo[1,...)
Affinity DataIC50: 3.53E+3nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223610BDBM50223610(3-bromo-N5-methyl-N7-(pyridin-3-ylmethyl)pyrazolo[...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223576BDBM50223576(3-ethynyl-5-phenyl-N-(pyridin-3-ylmethyl)pyrazolo[...)
Affinity DataIC50: 9.82E+3nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223570BDBM50223570(3-bromo-5-(2-fluorophenyl)-N-phenylpyrazolo[1,5-a]...)
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50223582BDBM50223582(N-benzyl-3-bromo-5-(2-fluorophenyl)pyrazolo[1,5-a]...)
Affinity DataIC50: 1.52E+4nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed