TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataKi: 0.560nMAssay Description:Displacement of [3H]NMS from rat muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]NMS from rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataKi: 12.7nMAssay Description:Displacement of [3H]NMS from rat muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataKi: 74.8nMAssay Description:Displacement of [3H]NMS from rat muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataKi: 85.7nMAssay Description:Displacement of [3H]NMS from rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataKi: 338nMAssay Description:Displacement of [3H]NMS from rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataKi: 445nMAssay Description:Displacement of [3H]NMS from rat muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 490nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 580nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 1.15E+3nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Antagonist activity at rat muscarinic M2 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 4.60E+3nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 5.10E+3nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 5.60E+3nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 7.60E+3nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 7.90E+3nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 1.88E+4nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 2.40E+4nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 2.90E+4nMAssay Description:Antagonist activity at rat muscarinic M2 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 5.20E+4nMAssay Description:Antagonist activity at rat muscarinic M2 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 6.60E+4nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: 7.00E+4nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M2 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M2 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair