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Found 64 Enz. Inhib. hit(s) with all data for entry = 50038257
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  0.560nMAssay Description:Displacement of [3H]NMS from rat muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]NMS from rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231845(CHEMBL255523 | N-(3-chloro-4-(4-ethylpiperazin-1-y...)
Affinity DataKi:  12.7nMAssay Description:Displacement of [3H]NMS from rat muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231845(CHEMBL255523 | N-(3-chloro-4-(4-ethylpiperazin-1-y...)
Affinity DataKi:  74.8nMAssay Description:Displacement of [3H]NMS from rat muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231845(CHEMBL255523 | N-(3-chloro-4-(4-ethylpiperazin-1-y...)
Affinity DataKi:  85.7nMAssay Description:Displacement of [3H]NMS from rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231845(CHEMBL255523 | N-(3-chloro-4-(4-ethylpiperazin-1-y...)
Affinity DataKi:  338nMAssay Description:Displacement of [3H]NMS from rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231845(CHEMBL255523 | N-(3-chloro-4-(4-ethylpiperazin-1-y...)
Affinity DataKi:  445nMAssay Description:Displacement of [3H]NMS from rat muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231845(CHEMBL255523 | N-(3-chloro-4-(4-ethylpiperazin-1-y...)
Affinity DataIC50:  440nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373835(CHEMBL256202)
Affinity DataIC50:  490nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373841(CHEMBL270580)
Affinity DataIC50:  580nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373834(CHEMBL255169)
Affinity DataIC50:  1.10E+3nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231845(CHEMBL255523 | N-(3-chloro-4-(4-ethylpiperazin-1-y...)
Affinity DataIC50:  1.10E+3nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373836(CHEMBL271704)
Affinity DataIC50:  1.15E+3nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231845(CHEMBL255523 | N-(3-chloro-4-(4-ethylpiperazin-1-y...)
Affinity DataIC50:  3.10E+3nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373832(CHEMBL429780)
Affinity DataIC50:  3.30E+3nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231845(CHEMBL255523 | N-(3-chloro-4-(4-ethylpiperazin-1-y...)
Affinity DataIC50:  3.50E+3nMAssay Description:Antagonist activity at rat muscarinic M2 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373837(CHEMBL429320)
Affinity DataIC50:  4.60E+3nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231856(CHEMBL271519 | N-(3-chloro-4-(4-ethylpiperazin-1-y...)
Affinity DataIC50:  5.00E+3nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373835(CHEMBL256202)
Affinity DataIC50:  5.10E+3nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373839(CHEMBL438706)
Affinity DataIC50:  5.60E+3nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373834(CHEMBL255169)
Affinity DataIC50:  7.60E+3nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373841(CHEMBL270580)
Affinity DataIC50:  7.90E+3nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373836(CHEMBL271704)
Affinity DataIC50:  1.30E+4nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373834(CHEMBL255169)
Affinity DataIC50:  1.80E+4nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373838(CHEMBL258335)
Affinity DataIC50:  1.88E+4nMAssay Description:Antagonist activity at rat muscarinic M1 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373836(CHEMBL271704)
Affinity DataIC50:  2.00E+4nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373836(CHEMBL271704)
Affinity DataIC50:  2.40E+4nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373836(CHEMBL271704)
Affinity DataIC50:  2.90E+4nMAssay Description:Antagonist activity at rat muscarinic M2 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373834(CHEMBL255169)
Affinity DataIC50:  5.20E+4nMAssay Description:Antagonist activity at rat muscarinic M2 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231856(CHEMBL271519 | N-(3-chloro-4-(4-ethylpiperazin-1-y...)
Affinity DataIC50:  6.60E+4nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373834(CHEMBL255169)
Affinity DataIC50:  7.00E+4nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373840(CHEMBL258281)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M2 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373833(CHEMBL404874)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373833(CHEMBL404874)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373832(CHEMBL429780)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231856(CHEMBL271519 | N-(3-chloro-4-(4-ethylpiperazin-1-y...)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373837(CHEMBL429320)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M3 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373833(CHEMBL404874)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231845(CHEMBL255523 | N-(3-chloro-4-(4-ethylpiperazin-1-y...)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373838(CHEMBL258335)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373839(CHEMBL438706)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373837(CHEMBL429320)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373840(CHEMBL258281)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373838(CHEMBL258335)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373832(CHEMBL429780)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373839(CHEMBL438706)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373837(CHEMBL429320)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373840(CHEMBL258281)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50373832(CHEMBL429780)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231856(CHEMBL271519 | N-(3-chloro-4-(4-ethylpiperazin-1-y...)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M2 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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