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Found 10 Enz. Inhib. hit(s) with all data for entry = 4675
TargetProto-oncogene tyrosine-protein kinase Src(Mus musculus (Mouse))
Ariad Pharmaceuticals

LigandPNGBDBM50318870(((4-(2-(cis-4-aminocyclohexyl)-9-ethyl-9H-purin-6-...)
Affinity DataIC50:  68nMAssay Description:2,6,9-Trisubstituted purines were evaluated for their src kinase inhibitory activities using an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetProto-oncogene tyrosine-protein kinase Src(Mus musculus (Mouse))
Ariad Pharmaceuticals

LigandPNGBDBM81725(2,6,9-Trisubstituted Purine, AP23517)
Affinity DataIC50:  73nMAssay Description:2,6,9-Trisubstituted purines were evaluated for their src kinase inhibitory activities using an ELISA assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Mus musculus (Mouse))
Ariad Pharmaceuticals

LigandPNGBDBM81723(2,6,9-Trisubstituted Purine, 10)
Affinity DataIC50:  101nMAssay Description:2,6,9-Trisubstituted purines were evaluated for their src kinase inhibitory activities using an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Mus musculus (Mouse))
Ariad Pharmaceuticals

LigandPNGBDBM81722(2,6,9-Trisubstituted Purine, 9)
Affinity DataIC50:  205nMAssay Description:2,6,9-Trisubstituted purines were evaluated for their src kinase inhibitory activities using an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Mus musculus (Mouse))
Ariad Pharmaceuticals

LigandPNGBDBM50318870(((4-(2-(cis-4-aminocyclohexyl)-9-ethyl-9H-purin-6-...)
Affinity DataIC50:  273nMAssay Description:2,6,9-Trisubstituted purines were evaluated for their src kinase inhibitory activities using an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetProto-oncogene tyrosine-protein kinase Src(Mus musculus (Mouse))
Ariad Pharmaceuticals

LigandPNGBDBM81718(2,6,9-Trisubstituted Purine, 4)
Affinity DataIC50:  665nMAssay Description:2,6,9-Trisubstituted purines were evaluated for their src kinase inhibitory activities using an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Mus musculus (Mouse))
Ariad Pharmaceuticals

LigandPNGBDBM81720(2,6,9-Trisubstituted Purine, 6)
Affinity DataIC50:  1.01E+3nMAssay Description:2,6,9-Trisubstituted purines were evaluated for their src kinase inhibitory activities using an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Mus musculus (Mouse))
Ariad Pharmaceuticals

LigandPNGBDBM81724(2,6,9-Trisubstituted Purine, 11)
Affinity DataIC50:  2.11E+3nMAssay Description:2,6,9-Trisubstituted purines were evaluated for their src kinase inhibitory activities using an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Mus musculus (Mouse))
Ariad Pharmaceuticals

LigandPNGBDBM81721(2,6,9-Trisubstituted Purine, 7)
Affinity DataIC50:  2.30E+3nMAssay Description:2,6,9-Trisubstituted purines were evaluated for their src kinase inhibitory activities using an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Mus musculus (Mouse))
Ariad Pharmaceuticals

LigandPNGBDBM81719(2,6,9-Trisubstituted Purine, 5)
Affinity DataIC50:  2.31E+3nMAssay Description:2,6,9-Trisubstituted purines were evaluated for their src kinase inhibitory activities using an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed