Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 2454
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM20732((4E,6Z,8S,9S,10E,12S,13R,14S,16R)-13-hydroxy-8,14,...)
Affinity DataIC50:  20nMpH: 7.3 T: 2°CAssay Description:Compounds were assayed over a threefold dilution series in a 96-well plate format to determine IC50 values. The reaction was allowed to proceed with ...More data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM20739(4-chloro-6-(5-{[2-(morpholin-4-yl)ethyl]amino}-1,2...)
Affinity DataIC50:  30nMpH: 7.3 T: 2°CAssay Description:Compounds were assayed over a threefold dilution series in a 96-well plate format to determine IC50 values. The reaction was allowed to proceed with ...More data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM20737(4-bromo-6-(5-{[2-(morpholin-4-yl)ethyl]amino}-1,2-...)
Affinity DataIC50:  40nMpH: 7.3 T: 2°CAssay Description:Compounds were assayed over a threefold dilution series in a 96-well plate format to determine IC50 values. The reaction was allowed to proceed with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM20734(4-chloro-6-(6-hydroxy-1,2-benzoxazol-3-yl)benzene-...)
Affinity DataIC50:  60nMpH: 7.3 T: 2°CAssay Description:Compounds were assayed over a threefold dilution series in a 96-well plate format to determine IC50 values. The reaction was allowed to proceed with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM20731(4-bromo-6-(6-hydroxy-1,2-benzoxazol-3-yl)benzene-1...)
Affinity DataIC50:  190nMpH: 7.3 T: 2°CAssay Description:Compounds were assayed over a threefold dilution series in a 96-well plate format to determine IC50 values. The reaction was allowed to proceed with ...More data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM20736(4-chloro-6-[5-(4-methylpiperazin-1-yl)-1,2-benzoxa...)
Affinity DataIC50:  800nMpH: 7.3 T: 2°CAssay Description:Compounds were assayed over a threefold dilution series in a 96-well plate format to determine IC50 values. The reaction was allowed to proceed with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM20733(4-(6-hydroxy-1,2-benzoxazol-3-yl)benzene-1,3-diol ...)
Affinity DataIC50:  1.52E+4nMpH: 7.3 T: 2°CAssay Description:Compounds were assayed over a threefold dilution series in a 96-well plate format to determine IC50 values. The reaction was allowed to proceed with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM20738(3-(5-chloro-2,4-dimethoxyphenyl)-N-[2-(morpholin-4...)
Affinity DataIC50: >2.00E+4nMpH: 7.3 T: 2°CAssay Description:Compounds were assayed over a threefold dilution series in a 96-well plate format to determine IC50 values. The reaction was allowed to proceed with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM20735(3-(5-chloro-2,4-dimethoxyphenyl)-6-methoxy-1,2-ben...)
Affinity DataIC50: >2.00E+4nMpH: 7.3 T: 2°CAssay Description:Compounds were assayed over a threefold dilution series in a 96-well plate format to determine IC50 values. The reaction was allowed to proceed with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed