Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50003964
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50067593BDBM50067593(CHEBI:44032 | Crixivan | Indinavir | L-735524 | MK...)
Affinity DataKi:  0.520nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478128BDBM50478128(CHEMBL442805)
Affinity DataKi:  2.30nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478106BDBM50478106(CHEMBL405316)
Affinity DataKi:  2.30nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478129BDBM50478129(CHEMBL270059)
Affinity DataKi:  2.40nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478108BDBM50478108(CHEMBL272832)
Affinity DataKi:  2.40nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13934BDBM13934(CGP 73547 | CHEMBL1163 | methyl N-[(1S)-1-{[(2S,3S...)
Affinity DataKi:  2.70nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478109BDBM50478109(CHEMBL539678)
Affinity DataKi:  2.80nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478118BDBM50478118(CHEMBL270135)
Affinity DataKi:  2.80nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478121BDBM50478121(CHEMBL271818)
Affinity DataKi:  2.90nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478110BDBM50478110(CHEMBL259895)
Affinity DataKi:  3.30nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478107BDBM50478107(CHEMBL429609)
Affinity DataKi:  3.30nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478116BDBM50478116(CHEMBL405041)
Affinity DataKi:  3.40nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478119BDBM50478119(CHEMBL405858)
Affinity DataKi:  3.5nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478125BDBM50478125(CHEMBL269874)
Affinity DataKi:  3.60nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478122BDBM50478122(CHEMBL406420)
Affinity DataKi:  3.60nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478103BDBM50478103(CHEMBL405019)
Affinity DataKi:  3.60nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478104BDBM50478104(CHEMBL272849)
Affinity DataKi:  4.5nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478115BDBM50478115(CHEMBL273031)
Affinity DataKi:  4.90nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478127BDBM50478127(CHEMBL273057)
Affinity DataKi:  5nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478105BDBM50478105(CHEMBL272848)
Affinity DataKi:  5.5nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478117BDBM50478117(CHEMBL259884)
Affinity DataKi:  5.70nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478111BDBM50478111(CHEMBL437606)
Affinity DataKi:  6.70nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478126BDBM50478126(CHEMBL442971)
Affinity DataKi:  6.80nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478113BDBM50478113(CHEMBL271756)
Affinity DataKi:  7.30nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478112BDBM50478112(CHEMBL407748)
Affinity DataKi:  10nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478120BDBM50478120(CHEMBL270080)
Affinity DataKi:  11nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478114BDBM50478114(CHEMBL405092)
Affinity DataKi:  24nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478101BDBM50478101(CHEMBL438010)
Affinity DataKi:  120nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478124BDBM50478124(CHEMBL405313)
Affinity DataKi:  190nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478123BDBM50478123(CHEMBL259039)
Affinity DataKi:  420nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
Uppsala University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50478102BDBM50478102(CHEMBL436861)
Affinity DataKi:  980nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2020
Entry Details Article
PubMed