Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50022310
TargetAngiotensin-converting enzyme 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21489BDBM21489(MLN4760 | (2S)-2-{[(1S)-1-carboxy-2-{1-[(3,5-dichl...)
Affinity DataIC50: 0.440nMAssay Description:Inhibition of ACE2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50233797BDBM50233797(DX-600 | CHEMBL436639)
Affinity DataIC50: 10nMAssay Description:Inhibition of ACE2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411606BDBM50411606(CHEMBL254282)
Affinity DataKi:  10nMAssay Description:Inhibition of human recombinant NEP by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411608BDBM50411608(CHEMBL400527)
Affinity DataKi:  12nMAssay Description:Inhibition of human recombinant NEP by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411598BDBM50411598(CHEMBL401397)
Affinity DataKi:  19nMAssay Description:Inhibition of human recombinant NEP by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411605BDBM50411605(CHEMBL252391)
Affinity DataKi:  27nMAssay Description:Inhibition of human recombinant NEP by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411613BDBM50411613(CHEMBL400526)
Affinity DataKi:  35nMAssay Description:Inhibition of human recombinant NEP by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411599BDBM50411599(CHEMBL254495)
Affinity DataKi:  37nMAssay Description:Inhibition of human recombinant NEP by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411607BDBM50411607(CHEMBL253428)
Affinity DataKi:  46nMAssay Description:Inhibition of human recombinant NEP by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411617BDBM50411617(CHEMBL253224)
Affinity DataKi:  75nMAssay Description:Inhibition of human recombinant NEP by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411603BDBM50411603(CHEMBL398771)
Affinity DataKi:  75nMAssay Description:Inhibition of human recombinant NEP by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411616BDBM50411616(CHEMBL252003)
Affinity DataKi:  79nMAssay Description:Inhibition of human recombinant NEP by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411610BDBM50411610(CHEMBL254493)
Affinity DataKi:  120nMAssay Description:Inhibition of human recombinant NEP by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411601BDBM50411601(CHEMBL254911)
Affinity DataKi:  180nMAssay Description:Inhibition of human recombinant NEP by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411611BDBM50411611(CHEMBL251804)
Affinity DataKi:  180nMAssay Description:Inhibition of human recombinant NEP by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411614BDBM50411614(CHEMBL398545)
Affinity DataKi:  190nMAssay Description:Inhibition of human recombinant NEP by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411612BDBM50411612(CHEMBL254703)
Affinity DataKi:  300nMAssay Description:Inhibition of human recombinant NEP by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411617BDBM50411617(CHEMBL253224)
Affinity DataKi:  350nMAssay Description:Inhibition of human recombinant CpA by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411613BDBM50411613(CHEMBL400526)
Affinity DataKi:  530nMAssay Description:Inhibition of human recombinant CpA by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411609BDBM50411609(CHEMBL251808)
Affinity DataKi:  640nMAssay Description:Inhibition of human recombinant NEP by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411602BDBM50411602(CHEMBL254900)
Affinity DataKi:  950nMAssay Description:Inhibition of human recombinant NEP by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411600BDBM50411600(CHEMBL251809)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of human recombinant NEP by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411610BDBM50411610(CHEMBL254493)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of human recombinant CpA by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411603BDBM50411603(CHEMBL398771)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition of human recombinant CpA by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411611BDBM50411611(CHEMBL251804)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of human recombinant CpA by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411609BDBM50411609(CHEMBL251808)
Affinity DataKi:  3.30E+3nMAssay Description:Inhibition of human recombinant CpA by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411608BDBM50411608(CHEMBL400527)
Affinity DataKi:  3.60E+3nMAssay Description:Inhibition of human recombinant CpA by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411600BDBM50411600(CHEMBL251809)
Affinity DataKi:  4.60E+3nMAssay Description:Inhibition of human recombinant CpA by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411612BDBM50411612(CHEMBL254703)
Affinity DataKi:  4.60E+3nMAssay Description:Inhibition of human recombinant CpA by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411599BDBM50411599(CHEMBL254495)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of human recombinant CpA by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411598BDBM50411598(CHEMBL401397)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of human recombinant CpA by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411615BDBM50411615(CHEMBL401086)
Affinity DataKi:  5.10E+3nMAssay Description:Inhibition of human recombinant NEP by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411607BDBM50411607(CHEMBL253428)
Affinity DataKi:  7.20E+3nMAssay Description:Inhibition of human recombinant CpA by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411606BDBM50411606(CHEMBL254282)
Affinity DataKi:  8.90E+3nMAssay Description:Inhibition of human recombinant CpA by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411614BDBM50411614(CHEMBL398545)
Affinity DataKi:  9.90E+3nMAssay Description:Inhibition of human recombinant CpA by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411604BDBM50411604(CHEMBL252009)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of human recombinant CpA by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411605BDBM50411605(CHEMBL252391)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of human recombinant CpA by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411602BDBM50411602(CHEMBL254900)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of human recombinant CpA by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411604BDBM50411604(CHEMBL252009)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of human recombinant NEP by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411616BDBM50411616(CHEMBL252003)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibition of human recombinant CpA by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411601BDBM50411601(CHEMBL254911)
Affinity DataKi:  1.60E+4nMAssay Description:Inhibition of human recombinant CpA by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50411615BDBM50411615(CHEMBL401086)
Affinity DataKi:  3.50E+4nMAssay Description:Inhibition of human recombinant CpA by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50233798BDBM50233798(N-(2-aminoethyl)-1-aziridine-ethanamine | CHEMBL39...)
Affinity DataIC50: 5.70E+4nMAssay Description:Inhibition of ACE2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 52871BDBM52871(CHEMBL252417 | (E)-3-[5-(5-chloro-2-methylphenyl)f...)
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibition of ACE2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed