Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50038360
TargetDelta-type opioid receptor(Homo sapiens (Human))
Westf£Lische Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50039029((+)-4-((alpha R)-((2S,5R)-4-allyl-2,5-dimethylpipe...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]deltorphine 2 from human delta opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Westf£Lische Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50375379(CHEMBL260519)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]naloxone from human mu opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Westf£Lische Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50375379(CHEMBL260519)
Affinity DataKi:  740nMAssay Description:Displacement of [3H]deltorphine 2 from human delta opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Westf£Lische Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50375376(CHEMBL260521)
Affinity DataKi:  890nMAssay Description:Displacement of [3H]C1-977 from human kappa opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Westf£Lische Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50375380(CHEMBL407728)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]C1-977 from human kappa opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Westf£Lische Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50375378(CHEMBL258791)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]C1-977 from human kappa opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Westf£Lische Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50375377(CHEMBL409266)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H]C1-977 from human kappa opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Westf£Lische Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50375377(CHEMBL409266)
Affinity DataKi:  5.70E+3nMAssay Description:Displacement of [3H]naloxone from human mu opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Westf£Lische Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50375380(CHEMBL407728)
Affinity DataKi:  6.32E+3nMAssay Description:Displacement of [3H]naloxone from human mu opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Westf£Lische Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50375376(CHEMBL260521)
Affinity DataKi:  6.80E+3nMAssay Description:Displacement of [3H]naloxone from human mu opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Westf£Lische Wilhelms-Universit£T

Curated by ChEMBL
LigandPNGBDBM50375378(CHEMBL258791)
Affinity DataKi:  7.30E+3nMAssay Description:Displacement of [3H]naloxone from human mu opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed