Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50038199
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373056(CHEMBL261163)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373048(CHEMBL184106)
Affinity DataIC50:  3.00E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373057(CHEMBL261162)
Affinity DataIC50:  3.60E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373047(CHEMBL260235)
Affinity DataIC50:  5.00E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373055(CHEMBL408369)
Affinity DataIC50:  5.00E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373052(CHEMBL404926)
Affinity DataIC50:  6.40E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373054(CHEMBL408296)
Affinity DataIC50:  7.20E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373053(CHEMBL260905)
Affinity DataIC50:  7.80E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373050(CHEMBL258584)
Affinity DataIC50:  9.40E+3nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373049(CHEMBL408121)
Affinity DataIC50:  1.30E+4nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandPNGBDBM50373051(CHEMBL404924)
Affinity DataIC50:  1.30E+4nMAssay Description:Antagonist activity at LuxR in Vibrio fischeri assessed as inhibition of N-3-oxos-hexanoyl-L-homoserine lactone induced luminescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed