Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50022519
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236065BDBM50236065((R)-3-(2-(1-(3-fluoro-5-methylphenyl)-2-methylprop...)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236057BDBM50236057((R)-3-(2-(1-(3-fluoro-4-methoxyphenyl)-2-methylpro...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236050BDBM50236050((R)-3-(2-(1-(3-cyano-5-fluorophenyl)propylamino)-3...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236066BDBM50236066((R)-3-(2-(1-(3,5-difluorophenyl)propylamino)-3,4-d...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236064BDBM50236064((R)-3-(2-(1-(3,5-difluorophenyl)-2-methylpropylami...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236068BDBM50236068((R)-3-(2-(1-(3-cyano-5-methylphenyl)propylamino)-3...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236059BDBM50236059((R)-3-(2-(1-(3-fluoro-5-methylphenyl)propylamino)-...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236062BDBM50236062((R)-2-hydroxy-N,N-dimethyl-3-(2-(2-methyl-1-(3-met...)
Affinity DataKi:  4.40nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236052BDBM50236052((R)-3-(2-(cyclopropyl(3,5-difluorophenyl)methylami...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236053BDBM50236053((R)-3-(3,4-dioxo-2-(1-phenylpropylamino)cyclobut-1...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50200885BDBM50200885((R)-3-(2-(1-(3-fluorophenyl)propylamino)-3,4-dioxo...)
Affinity DataIC50: 4.90nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50200885BDBM50200885((R)-3-(2-(1-(3-fluorophenyl)propylamino)-3,4-dioxo...)
Affinity DataIC50: 4.90nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236061BDBM50236061((R)-3-(2-(1-(3-fluoro-4-methoxyphenyl)propylamino)...)
Affinity DataKi:  5.20nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236056BDBM50236056(rac-3-(2-(1-(4-fluoro-3-methylphenyl)propylamino)-...)
Affinity DataKi:  6.10nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236053BDBM50236053((R)-3-(3,4-dioxo-2-(1-phenylpropylamino)cyclobut-1...)
Affinity DataIC50: 6.80nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236067BDBM50236067((R)-3-(2-(1-(3-fluoro-5-(trifluoromethyl)phenyl)pr...)
Affinity DataKi:  7.90nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236058BDBM50236058((R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(3-methyl-5-(tr...)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236063BDBM50236063((R)-3-(2-(1-(4-fluoro-3-methoxyphenyl)propylamino)...)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236054BDBM50236054((R)-3-(2-(1-(3-fluoro-5-(trifluoromethyl)phenyl)-2...)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236051BDBM50236051((R)-3-(2-(1-(3-fluoro-4-(trifluoromethyl)phenyl)-2...)
Affinity DataKi:  14nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236048BDBM50236048((R)-3-(2-(1-(4-fluoro-3-methoxyphenyl)-2-methylpro...)
Affinity DataKi:  16nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236049BDBM50236049((R)-3-(2-(1-(3-fluoro-4-(trifluoromethyl)phenyl)pr...)
Affinity DataKi:  19nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236055BDBM50236055(rac-3-(2-(1-(3,4-difluorophenyl)propylamino)-3,4-d...)
Affinity DataKi:  28nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Pharmacopeia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236060BDBM50236060((R)-3-(2-(1-(4-fluoro-3-(trifluoromethyl)phenyl)pr...)
Affinity DataKi:  39nMAssay Description:Displacement of [125I]IL8 from human CXCR2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed