Compile Data Set for Download or QSAR
maximum 50k data
Found 40 Enz. Inhib. hit(s) with all data for entry = 50022549
TargetMitogen-activated protein kinase 11(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236473((R)-2-(sec-butylamino)-N-(2-methyl-5-(methylcarbam...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of human p38betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236476(CHEMBL255482 | N-(5-(ethylcarbamoyl)-2-methylpheny...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236483((S)-2-(sec-butylamino)-N-(2-methyl-5-(methylcarbam...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236490(CHEMBL257995 | N-(5-carbamoyl-2-methylphenyl)-2-(i...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236474(CHEMBL255698 | N-(5-(ethylcarbamoyl)-2-methylpheny...)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236473((R)-2-(sec-butylamino)-N-(2-methyl-5-(methylcarbam...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236475(2-(isopropylamino)-N-(2-methyl-5-(methylcarbamoyl)...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236487(2-(isopropylamino)-N-(5-(isoxazol-3-ylcarbamoyl)-2...)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236488(CHEMBL257994 | N-(5-carbamoyl-2-methylphenyl)-2-(p...)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236478(CHEMBL255288 | N-(5-((1H-pyrazol-5-yl)carbamoyl)-2...)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236480(CHEMBL257996 | N-(2-methyl-5-(methylcarbamoyl)phen...)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236485(2-(isopropylamino)-N-(2-methyl-5-((1-methyl-1H-pyr...)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236482(CHEMBL403141 | N-(2-chloro-6-methylphenyl)-2-(isop...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236477(2-(2-methoxyethylamino)-N-(2-methyl-5-(methylcarba...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236486(CHEMBL255254 | N-(2-chloro-6-methylphenyl)-2-(prop...)
Affinity DataIC50:  28nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236479(CHEMBL254169 | N-ethyl-3-(2-(isopropylamino)-6-oxo...)
Affinity DataIC50:  34nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236484(CHEMBL255428 | N-(2-chloro-6-methylphenyl)-2-(cycl...)
Affinity DataIC50:  36nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236481(CHEMBL258403 | N-(2-chloro-6-methylphenyl)-2-(cycl...)
Affinity DataIC50:  39nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236471(3-(2-(cyclopentylamino)-6-oxo-3a,4,6,6a-tetrahydro...)
Affinity DataIC50:  53nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50156469(2-Phenylamino-thiazole-5-carboxylic acid (2-chloro...)
Affinity DataIC50:  62nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236495(3-(2-(isopropylamino)-6-oxo-4H-pyrrolo[3,4-d]thiaz...)
Affinity DataIC50:  110nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236491(3-(2-(cyclopentylamino)-6-oxo-4H-pyrrolo[3,4-d]thi...)
Affinity DataIC50:  110nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236472(CHEMBL404446 | N-(5-(ethylcarbamoyl)-2-methylpheny...)
Affinity DataIC50:  130nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236481(CHEMBL258403 | N-(2-chloro-6-methylphenyl)-2-(cycl...)
Affinity DataIC50:  140nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236493(CHEMBL403140 | N-(2-chloro-6-methylphenyl)-2-(ethy...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236494(CHEMBL254168 | N-ethyl-4-methyl-3-(6-oxo-2-(propyl...)
Affinity DataIC50:  160nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236492(CHEMBL255719 | N,4-dimethyl-3-(6-oxo-2-(propylamin...)
Affinity DataIC50:  270nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236489(2-(ethylamino)-N-(5-(ethylcarbamoyl)-2-methylpheny...)
Affinity DataIC50:  330nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236487(2-(isopropylamino)-N-(5-(isoxazol-3-ylcarbamoyl)-2...)
Affinity DataIC50:  380nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236476(CHEMBL255482 | N-(5-(ethylcarbamoyl)-2-methylpheny...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236484(CHEMBL255428 | N-(2-chloro-6-methylphenyl)-2-(cycl...)
Affinity DataIC50:  3.31E+3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236480(CHEMBL257996 | N-(2-methyl-5-(methylcarbamoyl)phen...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236485(2-(isopropylamino)-N-(2-methyl-5-((1-methyl-1H-pyr...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236473((R)-2-(sec-butylamino)-N-(2-methyl-5-(methylcarbam...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 12(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236473((R)-2-(sec-butylamino)-N-(2-methyl-5-(methylcarbam...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human p38gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 13(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236473((R)-2-(sec-butylamino)-N-(2-methyl-5-(methylcarbam...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human p38deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236483((S)-2-(sec-butylamino)-N-(2-methyl-5-(methylcarbam...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236490(CHEMBL257995 | N-(5-carbamoyl-2-methylphenyl)-2-(i...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236474(CHEMBL255698 | N-(5-(ethylcarbamoyl)-2-methylpheny...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236475(2-(isopropylamino)-N-(2-methyl-5-(methylcarbamoyl)...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed