Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 4676
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital

LigandPNGBDBM3294(4-Anilinoquinazoline deriv. 45 | 4-N-(3-bromopheny...)
Affinity DataIC50:  44nMT: 2°CAssay Description:EGFR kinase assay was perform using Nunc MaxiSorp purchased from Nalge Nunc Interantional.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital

LigandPNGBDBM81727(Bis-quinazolinotriazene, 5b)
Affinity DataIC50:  120nMT: 2°CAssay Description:EGFR kinase assay was perform using Nunc MaxiSorp purchased from Nalge Nunc Interantional.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital

LigandPNGBDBM81728(Bis-quinazolinotriazene, 5c)
Affinity DataIC50:  150nMT: 2°CAssay Description:EGFR kinase assay was perform using Nunc MaxiSorp purchased from Nalge Nunc Interantional.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital

LigandPNGBDBM50133382(Anilinoquinazoline, 4c | CHEMBL343352 | N*4*-(3-Ch...)
Affinity DataIC50:  200nMT: 2°CAssay Description:EGFR kinase assay was perform using Nunc MaxiSorp purchased from Nalge Nunc Interantional.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital

LigandPNGBDBM81726(Bis-quinazolinotriazene, 5a)
Affinity DataIC50:  950nMT: 2°CAssay Description:EGFR kinase assay was perform using Nunc MaxiSorp purchased from Nalge Nunc Interantional.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital

LigandPNGBDBM50133384(Anilinoquinazoline, 4a | CHEMBL336113 | N*4*-m-Tol...)
Affinity DataIC50:  1.00E+3nMT: 2°CAssay Description:EGFR kinase assay was perform using Nunc MaxiSorp purchased from Nalge Nunc Interantional.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed