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Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50038832
TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266372(CHEMBL451321 | metaglidasen)
Affinity DataIC50:  220nMAssay Description:Antagonist activity at human PPARgamma receptor expressed in Saccharomyces cerevisiae AH109 co-transfected with mouse CBP assessed as inhibition of r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266362((Z)-N-(3-allyl-5-nitrothiazol-2(3H)-ylidene)pivala...)
Affinity DataIC50:  820nMAssay Description:Antagonist activity at human PPARgamma receptor expressed in Saccharomyces cerevisiae AH109 co-transfected with mouse CBP assessed as inhibition of r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266373(2-chloro-5-nitro-N-(pyridin-4-yl)benzamide | CHEMB...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at human PPARgamma receptor expressed in Saccharomyces cerevisiae AH109 co-transfected with mouse CBP assessed as inhibition of r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50837(MLS000099571 | N-[2-(4-fluorophenyl)ethyl]-4-metho...)
Affinity DataIC50:  3.30E+3nMAssay Description:Antagonist activity at human PPARgamma receptor expressed in Saccharomyces cerevisiae AH109 co-transfected with mouse CBP assessed as inhibition of r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266632(CHEMBL476008 | L-Tryptophan-L-aspartic acid)
Affinity DataIC50:  5.20E+3nMAssay Description:Antagonist activity at human PPARgamma receptor expressed in Saccharomyces cerevisiae AH109 co-transfected with mouse CBP assessed as inhibition of r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50240464((S)-2-((S)-2-amino-3-(1H-indol-3-yl)propanamido)pe...)
Affinity DataIC50:  8.67E+3nMAssay Description:Antagonist activity at human PPARgamma receptor expressed in Saccharomyces cerevisiae AH109 co-transfected with mouse CBP assessed as inhibition of r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266633(CHEMBL515773 | L-Tryptophan-L-2-aminoadipic acid)
Affinity DataIC50:  1.51E+4nMAssay Description:Antagonist activity at human PPARgamma receptor expressed in Saccharomyces cerevisiae AH109 co-transfected with mouse CBP assessed as inhibition of r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266680(CHEMBL477417 | L-Tryptophan-L-arginine)
Affinity DataIC50:  1.54E+4nMAssay Description:Antagonist activity at human PPARgamma receptor expressed in Saccharomyces cerevisiae AH109 co-transfected with mouse CBP assessed as inhibition of r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266679(CHEMBL513911 | L-Tryptophan-L-asparagine)
Affinity DataIC50:  1.84E+4nMAssay Description:Antagonist activity at human PPARgamma receptor expressed in Saccharomyces cerevisiae AH109 co-transfected with mouse CBP assessed as inhibition of r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266654(CHEMBL476173 | L-Tryptophan-L-glutamine)
Affinity DataIC50:  1.87E+4nMAssay Description:Antagonist activity at human PPARgamma receptor expressed in Saccharomyces cerevisiae AH109 co-transfected with mouse CBP assessed as inhibition of r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266681(CHEMBL477627 | L-Tryptophan-L-leucine)
Affinity DataIC50:  2.58E+4nMAssay Description:Antagonist activity at human PPARgamma receptor expressed in Saccharomyces cerevisiae AH109 co-transfected with mouse CBP assessed as inhibition of r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50266371(CHEMBL456071 | HALOFENATE)
Affinity DataIC50:  4.00E+4nMAssay Description:Antagonist activity at human PPARgamma receptor expressed in Saccharomyces cerevisiae AH109 co-transfected with mouse CBP assessed as inhibition of r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50241439(2,2'-(4,4'-(propane-2,2-diyl)bis(4,1-phenylene))bi...)
Affinity DataIC50:  1.00E+5nMAssay Description:Antagonist activity at human PPARgamma receptor expressed in Saccharomyces cerevisiae AH109 co-transfected with mouse CBP assessed as inhibition of r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Human)
Graduate School of The Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50240444((4-chlorophenyl)(dimethoxyphosphoryl)methyl dimeth...)
Affinity DataIC50:  1.40E+5nMAssay Description:Antagonist activity at human PPARgamma receptor expressed in Saccharomyces cerevisiae AH109 co-transfected with mouse CBP assessed as inhibition of r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed