Compile Data Set for Download or QSAR
maximum 50k data
Found 77 Enz. Inhib. hit(s) with all data for entry = 50025827
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataKi:  13nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247371(CHEMBL454923 | N-benzyl-1-(2-chloro-2-phenylethyl)...)
Affinity DataKi:  100nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247366(CHEMBL454119 | N-butyl-1-(2-chloro-2-(4-fluorophen...)
Affinity DataKi:  110nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247253(CHEMBL473726 | N4-benzyl-1-(2-chloro-2-phenylethyl...)
Affinity DataKi:  160nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247202(CHEMBL473516 | N-benzyl-1-(2-bromo-2-phenylethyl)-...)
Affinity DataKi:  190nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247200(1-(2-chloro-2-(4-fluorophenyl)ethyl)-6-(methylthio...)
Affinity DataKi:  200nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247248(1-(2-chloro-2-(4-fluorophenyl)ethyl)-N-(3-fluoroph...)
Affinity DataKi:  210nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247248(1-(2-chloro-2-(4-fluorophenyl)ethyl)-N-(3-fluoroph...)
Affinity DataKi:  220nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247202(CHEMBL473516 | N-benzyl-1-(2-bromo-2-phenylethyl)-...)
Affinity DataKi:  220nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247198(1-(2-chloro-2-(4-fluorophenyl)ethyl)-N-(4-fluorobe...)
Affinity DataKi:  220nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247368(1-(2-chloro-2-phenylethyl)-N-propyl-6-(propylthio)...)
Affinity DataKi:  250nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247203(1-(2-bromo-2-phenylethyl)-6-(methylthio)-N-pheneth...)
Affinity DataKi:  270nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247255(1-(2-chloro-2-phenylethyl)-N,N-dimethyl-4-morpholi...)
Affinity DataKi:  280nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247370(1-(2-chloro-2-phenylethyl)-N,N-diethyl-6-(propylth...)
Affinity DataKi:  280nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247199(1-(2-chloro-2-(4-fluorophenyl)ethyl)-N-(2-fluorobe...)
Affinity DataKi:  300nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50142885(Benzyl-[1-(2-chloro-2-phenyl-ethyl)-6-methylsulfan...)
Affinity DataKi:  300nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247251(1-(2-chloro-2-(4-chlorophenyl)ethyl)-N,N-diethyl-6...)
Affinity DataKi:  300nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247198(1-(2-chloro-2-(4-fluorophenyl)ethyl)-N-(4-fluorobe...)
Affinity DataKi:  310nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247386(1-(2-bromo-2-phenylethyl)-N-butyl-6-(methylthio)-1...)
Affinity DataKi:  320nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247389(1-(2-bromo-2-phenylethyl)-6-(methylthio)-4-(piperi...)
Affinity DataKi:  320nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247254(1-(2-chloro-2-phenylethyl)-N6,N6-dimethyl-N4-propy...)
Affinity DataKi:  320nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247367(1-(2-chloro-2-phenylethyl)-N,N-diethyl-6-(ethylthi...)
Affinity DataKi:  330nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247199(1-(2-chloro-2-(4-fluorophenyl)ethyl)-N-(2-fluorobe...)
Affinity DataKi:  340nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247250(CHEMBL475337 | N-butyl-1-(2-chloro-2-(4-chlorophen...)
Affinity DataKi:  390nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247364(1-(2-chloro-2-phenylethyl)-N-(2-fluorophenethyl)-6...)
Affinity DataKi:  400nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224381(1-(2-chloro-2-phenylethyl)-N-(3-fluorophenyl)-6-(m...)
Affinity DataKi:  400nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224385(1-(2-chloro-2-phenylethyl)-6-(methylthio)-N-phenyl...)
Affinity DataKi:  400nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50145415(1-(2-chloro-2-phenylethyl)-N,N-diethyl-6-(methylth...)
Affinity DataKi:  400nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247249(1-(2-chloro-2-(4-chlorophenyl)ethyl)-6-(methylthio...)
Affinity DataKi:  400nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247252(4-(1-(2-chloro-2-(4-chlorophenyl)ethyl)-6-(methylt...)
Affinity DataKi:  500nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50145415(1-(2-chloro-2-phenylethyl)-N,N-diethyl-6-(methylth...)
Affinity DataKi:  500nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50241420(4-amino-5-(4-chlorophenyl)-7-(t-butyl)pyrazolo[ 3,...)
Affinity DataKi:  500nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247371(CHEMBL454923 | N-benzyl-1-(2-chloro-2-phenylethyl)...)
Affinity DataKi:  510nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247369(CHEMBL454922 | N-butyl-1-(2-chloro-2-phenylethyl)-...)
Affinity DataKi:  520nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50241420(4-amino-5-(4-chlorophenyl)-7-(t-butyl)pyrazolo[ 3,...)
Affinity DataKi:  520nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247387(1-(2-bromo-2-phenylethyl)-N-(2-ethoxyethyl)-6-(met...)
Affinity DataKi:  550nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247365(1-(2-chloro-2-(4-fluorophenyl)ethyl)-6-(methylthio...)
Affinity DataKi:  570nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50142880(1-(2-chloro-2-phenylethyl)-6-(methylthio)-N-phenet...)
Affinity DataKi:  700nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247386(1-(2-bromo-2-phenylethyl)-N-butyl-6-(methylthio)-1...)
Affinity DataKi:  810nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247389(1-(2-bromo-2-phenylethyl)-6-(methylthio)-4-(piperi...)
Affinity DataKi:  880nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247385(1-(2-bromo-2-phenylethyl)-6-(methylthio)-N-propyl-...)
Affinity DataKi:  880nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247201(4-(1-(2-bromo-2-phenylethyl)-6-(methylthio)-1H-pyr...)
Affinity DataKi:  970nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247197(4-(1-(2-chloro-2-(4-fluorophenyl)ethyl)-6-(methylt...)
Affinity DataKi:  970nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224385(1-(2-chloro-2-phenylethyl)-6-(methylthio)-N-phenyl...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50142889(Butyl-[1-(2-chloro-2-phenyl-ethyl)-6-methylsulfany...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247249(1-(2-chloro-2-(4-chlorophenyl)ethyl)-6-(methylthio...)
Affinity DataKi:  1.32E+3nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224381(1-(2-chloro-2-phenylethyl)-N-(3-fluorophenyl)-6-(m...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247388(1-(2-bromo-2-phenylethyl)-6-(methylthio)-4-(pyrrol...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50142883(1-(2-chloro-2-phenylethyl)-N-(2-ethoxyethyl)-6-(me...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of human recombinant Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247250(CHEMBL475337 | N-butyl-1-(2-chloro-2-(4-chlorophen...)
Affinity DataKi:  1.53E+3nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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