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Found 61 Enz. Inhib. hit(s) with all data for entry = 50038425
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354515(CHEMBL261719)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354492(CHEMBL260994)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354521(CHEMBL408976)
Affinity DataKi:  0.410nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354506(CHEMBL260872)
Affinity DataKi:  0.430nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354522(CHEMBL261209)
Affinity DataKi:  0.490nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376328(CHEMBL406414)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354503(CHEMBL259087)
Affinity DataKi:  0.630nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376339(CHEMBL259086)
Affinity DataKi:  0.660nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376324(CHEMBL259549)
Affinity DataKi:  0.670nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354493(CHEMBL409662)
Affinity DataKi:  0.790nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376327(CHEMBL410226)
Affinity DataKi:  1.02nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354497(CHEMBL410225)
Affinity DataKi:  1.19nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376336(CHEMBL262068)
Affinity DataKi:  1.24nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376342(CHEMBL258496)
Affinity DataKi:  1.45nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376332(CHEMBL259216)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376340(CHEMBL408191)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376333(CHEMBL408450)
Affinity DataKi:  1.96nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376335(CHEMBL410628)
Affinity DataKi:  2.07nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354491(CHEMBL259550)
Affinity DataKi:  2.11nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376330(CHEMBL260762)
Affinity DataKi:  2.55nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354514(CHEMBL259010)
Affinity DataKi:  2.81nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376331(CHEMBL408426)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354513(CHEMBL269083)
Affinity DataKi:  3.72nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376326(CHEMBL410128)
Affinity DataKi:  4.31nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376337(CHEMBL259215)
Affinity DataKi:  4.75nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354523(CHEMBL407412)
Affinity DataKi:  5.11nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354496(CHEMBL258537)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354524(CHEMBL265927)
Affinity DataKi:  5.38nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376322(CHEMBL260761)
Affinity DataKi:  5.97nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376334(CHEMBL408451)
Affinity DataKi:  6.57nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354512(CHEMBL260551)
Affinity DataKi:  6.99nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376325(CHEMBL407263)
Affinity DataKi:  7.65nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376338(CHEMBL411919)
Affinity DataKi:  8.27nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354519(CHEMBL261009)
Affinity DataKi:  9.07nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376323(CHEMBL259009)
Affinity DataKi:  9.46nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354511(CHEMBL260870)
Affinity DataKi:  10.1nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354492(CHEMBL260994)
Affinity DataKi:  17.5nMAssay Description:Inhibition of 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354493(CHEMBL409662)
Affinity DataKi:  19.4nMAssay Description:Inhibition of 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354525(CHEMBL411663)
Affinity DataKi:  20nMAssay Description:Inhibition of adrenergic alpha-1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376321(CHEMBL412143)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376329(CHEMBL258593)
Affinity DataKi:  25.4nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50376341(CHEMBL408429)
Affinity DataKi:  33.4nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354492(CHEMBL260994)
Affinity DataKi:  42nMAssay Description:Inhibition of adrenergic alpha-1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354525(CHEMBL411663)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354525(CHEMBL411663)
Affinity DataKi:  55nMAssay Description:Inhibition of 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354493(CHEMBL409662)
Affinity DataKi:  71.3nMAssay Description:Inhibition of adrenergic alpha-1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354525(CHEMBL411663)
Affinity DataKi:  150nMAssay Description:Inhibition of 5HT1A receptor in rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354493(CHEMBL409662)
Affinity DataKi:  187nMAssay Description:Inhibition of 5HT6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354525(CHEMBL411663)
Affinity DataKi:  330nMAssay Description:Inhibition of dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50354493(CHEMBL409662)
Affinity DataKi:  358nMAssay Description:Inhibition of 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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