Compile Data Set for Download or QSAR
maximum 50k data
Found 59 Enz. Inhib. hit(s) with all data for entry = 50025870
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247269((2S,4S)-4-(3,4,5-Trimethoxybenzamido)-1-acetyl-Nhy...)
Affinity DataIC50:  1nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247519((2S,4S)-1-Acetyl-4-(cinnamamido)-N-hydroxypyrrolid...)
Affinity DataIC50:  4nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247270(CHEMBL472906 | N-((3S,5S)-5-(Hydroxycarbamoyl)-1-a...)
Affinity DataIC50:  5nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247539(CHEMBL472915 | N-((3S,5S)-1-((E)-3-(3,4-dimethoxyp...)
Affinity DataIC50:  9nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247521((2S,4S)-1-(3-(3,4-Dimethoxyphenyl)propanoyl)-4-(ci...)
Affinity DataIC50:  11nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247520(CHEMBL514309 | N-((3S,5S)-5-(Hydroxycarbamoyl)-1-(...)
Affinity DataIC50:  12nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247522((2S,4S)-4-(3,4,5-trimethoxybenzamido)-1-acetylpyrr...)
Affinity DataIC50:  16nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247218((2S,4S)-Methyl 1-acetyl-4-(cinnamamido)pyrrolidine...)
Affinity DataIC50:  100nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247517((2S,4S)-Methyl 4-(3,4,5-trimethoxybenzamido)-1-ace...)
Affinity DataIC50:  100nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247523(CHEMBL473732 | methyl 2-((2S,4S)-4-(3,4,5-trimetho...)
Affinity DataIC50:  109nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247265((3R,5S)-5-(methoxycarbonyl)-1-acetylpyrrolidin-3-y...)
Affinity DataIC50:  300nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247219((2S,4S)-Methyl 4-((E)-3-(3,4-dimethoxyphenyl)acryl...)
Affinity DataIC50:  800nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247518((2S,4S)-Methyl 1-acetyl-4-(nicotinamido)pyrrolidin...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247492((3R,5S)-5-(methoxycarbonyl)-1-((E)-3-(3,4-dimethox...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247495((2S,4S)-methyl 1-acetyl-4-aminopyrrolidine-2-carbo...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247268((2S,4S)-Methyl 1-(3-(3,4-dimethoxyphenyl)propanoyl...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247263((2S,4R)-methyl 1-acetyl-4-hydroxypyrrolidine-2-car...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247497((2S,4S)-methyl 1-(3-(3,4-dimethoxyphenyl)propanoyl...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247217((2S,4S)-Methyl 1-acetyl-4-(pyrazine-2-carboxamido)...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247267((2S,4S)-Methyl 1-(3-(3,4-dimethoxyphenyl)propanoyl...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247216((2S,4S)-Methyl 1-acetyl-4-(isonicotinamido)pyrroli...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247493((2S,4S)-methyl 1-acetyl-4-azidopyrrolidine-2-carbo...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247513((2S,4S)-Methyl 1-acetyl-4-(benzamido)pyrrolidine-2...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247264((2S,4R)-methyl 4-hydroxy-1-((E)-3-(3,4-dimethoxyph...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247266((2S,4S)-Methyl 1-((E)-3-(3,4-dimethoxyphenyl)acryl...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247494((2S,4S)-methyl 4-azido-1-((E)-3-(3,4-dimethoxyphen...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247514((2S,4S)-Methyl 4-(4-chlorobenzamido)-1-acetylpyrro...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247516((2S,4S)-Methyl 4-(4-nitrobenzamido)-1-acetylpyrrol...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247515((2S,4S)-Methyl 4-(4-bromobenzamido)-1-acetylpyrrol...)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of MMP2 (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247495((2S,4S)-methyl 1-acetyl-4-aminopyrrolidine-2-carbo...)
Affinity DataIC50:  2.41E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247270(CHEMBL472906 | N-((3S,5S)-5-(Hydroxycarbamoyl)-1-a...)
Affinity DataIC50:  2.98E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247265((3R,5S)-5-(methoxycarbonyl)-1-acetylpyrrolidin-3-y...)
Affinity DataIC50:  3.04E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247269((2S,4S)-4-(3,4,5-Trimethoxybenzamido)-1-acetyl-Nhy...)
Affinity DataIC50:  3.35E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247263((2S,4R)-methyl 1-acetyl-4-hydroxypyrrolidine-2-car...)
Affinity DataIC50:  3.86E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247492((3R,5S)-5-(methoxycarbonyl)-1-((E)-3-(3,4-dimethox...)
Affinity DataIC50:  4.66E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247522((2S,4S)-4-(3,4,5-trimethoxybenzamido)-1-acetylpyrr...)
Affinity DataIC50:  5.14E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247519((2S,4S)-1-Acetyl-4-(cinnamamido)-N-hydroxypyrrolid...)
Affinity DataIC50:  5.61E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247520(CHEMBL514309 | N-((3S,5S)-5-(Hydroxycarbamoyl)-1-(...)
Affinity DataIC50:  6.22E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247497((2S,4S)-methyl 1-(3-(3,4-dimethoxyphenyl)propanoyl...)
Affinity DataIC50:  6.84E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247496((2S,4S)-methyl 4-amino-1-((E)-3-(3,4-dimethoxyphen...)
Affinity DataIC50:  7.06E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247494((2S,4S)-methyl 4-azido-1-((E)-3-(3,4-dimethoxyphen...)
Affinity DataIC50:  7.13E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247516((2S,4S)-Methyl 4-(4-nitrobenzamido)-1-acetylpyrrol...)
Affinity DataIC50:  7.23E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247493((2S,4S)-methyl 1-acetyl-4-azidopyrrolidine-2-carbo...)
Affinity DataIC50:  7.37E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247216((2S,4S)-Methyl 1-acetyl-4-(isonicotinamido)pyrroli...)
Affinity DataIC50:  7.48E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247518((2S,4S)-Methyl 1-acetyl-4-(nicotinamido)pyrrolidin...)
Affinity DataIC50:  7.84E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247264((2S,4R)-methyl 4-hydroxy-1-((E)-3-(3,4-dimethoxyph...)
Affinity DataIC50:  8.18E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247217((2S,4S)-Methyl 1-acetyl-4-(pyrazine-2-carboxamido)...)
Affinity DataIC50:  8.26E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247521((2S,4S)-1-(3-(3,4-Dimethoxyphenyl)propanoyl)-4-(ci...)
Affinity DataIC50:  9.66E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247517((2S,4S)-Methyl 4-(3,4,5-trimethoxybenzamido)-1-ace...)
Affinity DataIC50:  9.84E+4nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247523(CHEMBL473732 | methyl 2-((2S,4S)-4-(3,4,5-trimetho...)
Affinity DataIC50:  1.22E+5nMAssay Description:Inhibition of aminopeptidase N (unknown origin) by microtiter plate fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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