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Found 18 Enz. Inhib. hit(s) with all data for entry = 50026096
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Wisconsin-La Crosse

Curated by ChEMBL
LigandPNGBDBM50052337(2-(8-bromo-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']d...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Wisconsin-La Crosse

Curated by ChEMBL
LigandPNGBDBM50271489(1-(4-Bromo-7,8-dihydro-6H-furo[2,3-g]chromen-9-yl)...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Wisconsin-La Crosse

Curated by ChEMBL
LigandPNGBDBM50271484(2-(10-Bromo-2,3,4,7,8,9-hexahydro-pyrano[2,3-g]chr...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Wisconsin-La Crosse

Curated by ChEMBL
LigandPNGBDBM50271486(1-(4-Bromo-3,6,7,8-tetrahydro-2H-furo[2,3-g]chrome...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Wisconsin-La Crosse

Curated by ChEMBL
LigandPNGBDBM50271483(2-(10-Bromo-2,3,4,7,8,9-hexahydro-pyrano[2,3-g]chr...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Wisconsin-La Crosse

Curated by ChEMBL
LigandPNGBDBM50271488(1-(9-Bromo-3,6,7,8-tetrahydro-2H-furo[2,3-g]chrome...)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Wisconsin-La Crosse

Curated by ChEMBL
LigandPNGBDBM50271487(2-(9-Bromo-3,6,7,8-tetrahydro-2H-furo[2,3-g]chrome...)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Wisconsin-La Crosse

Curated by ChEMBL
LigandPNGBDBM50271485(2-(4-Bromo-3,6,7,8-tetrahydro-2H-furo[2,3-g]chrome...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Wisconsin-La Crosse

Curated by ChEMBL
LigandPNGBDBM50005257((+)-2-(4-Bromo-2,5-dimethoxy-phenyl)-1-methyl-ethy...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Wisconsin-La Crosse

Curated by ChEMBL
LigandPNGBDBM50271483(2-(10-Bromo-2,3,4,7,8,9-hexahydro-pyrano[2,3-g]chr...)
Affinity DataEC50:  241nMAssay Description:Agonist activity at rat 5HT2A receptor expressed in mouse NIH3T3 cells assessed as stimulation of inositol phosphate accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Wisconsin-La Crosse

Curated by ChEMBL
LigandPNGBDBM50271484(2-(10-Bromo-2,3,4,7,8,9-hexahydro-pyrano[2,3-g]chr...)
Affinity DataEC50:  258nMAssay Description:Agonist activity at rat 5HT2A receptor expressed in mouse NIH3T3 cells assessed as stimulation of inositol phosphate accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Wisconsin-La Crosse

Curated by ChEMBL
LigandPNGBDBM50271485(2-(4-Bromo-3,6,7,8-tetrahydro-2H-furo[2,3-g]chrome...)
Affinity DataEC50:  9.40nMAssay Description:Agonist activity at rat 5HT2A receptor expressed in mouse NIH3T3 cells assessed as stimulation of inositol phosphate accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Wisconsin-La Crosse

Curated by ChEMBL
LigandPNGBDBM50271486(1-(4-Bromo-3,6,7,8-tetrahydro-2H-furo[2,3-g]chrome...)
Affinity DataEC50:  19nMAssay Description:Agonist activity at rat 5HT2A receptor expressed in mouse NIH3T3 cells assessed as stimulation of inositol phosphate accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Wisconsin-La Crosse

Curated by ChEMBL
LigandPNGBDBM50271487(2-(9-Bromo-3,6,7,8-tetrahydro-2H-furo[2,3-g]chrome...)
Affinity DataEC50:  146nMAssay Description:Agonist activity at rat 5HT2A receptor expressed in mouse NIH3T3 cells assessed as stimulation of inositol phosphate accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Wisconsin-La Crosse

Curated by ChEMBL
LigandPNGBDBM50271488(1-(9-Bromo-3,6,7,8-tetrahydro-2H-furo[2,3-g]chrome...)
Affinity DataEC50:  78nMAssay Description:Agonist activity at rat 5HT2A receptor expressed in mouse NIH3T3 cells assessed as stimulation of inositol phosphate accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Wisconsin-La Crosse

Curated by ChEMBL
LigandPNGBDBM50271489(1-(4-Bromo-7,8-dihydro-6H-furo[2,3-g]chromen-9-yl)...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at rat 5HT2A receptor expressed in mouse NIH3T3 cells assessed as stimulation of inositol phosphate accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Wisconsin-La Crosse

Curated by ChEMBL
LigandPNGBDBM50052337(2-(8-bromo-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']d...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at rat 5HT2A receptor expressed in mouse NIH3T3 cells assessed as stimulation of inositol phosphate accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Wisconsin-La Crosse

Curated by ChEMBL
LigandPNGBDBM50005257((+)-2-(4-Bromo-2,5-dimethoxy-phenyl)-1-methyl-ethy...)
Affinity DataEC50:  22nMAssay Description:Agonist activity at rat 5HT2A receptor expressed in mouse NIH3T3 cells assessed as stimulation of inositol phosphate accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed