Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 3585
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University of Pennsylvania

LigandPNGBDBM36523(DW12)
Affinity DataIC50:  1.40nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization-based kinase in vitro assay using human PI3K alpha purchased from Echelon Biosciences and p110 alpha/p85 alpha from Upstate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University of Pennsylvania

LigandPNGBDBM36525(EAd125)
Affinity DataIC50:  40nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization-based kinase in vitro assay using human PI3K alpha purchased from Echelon Biosciences and p110 alpha/p85 alpha from Upstate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University of Pennsylvania

LigandPNGBDBM36522(HB12)
Affinity DataIC50:  50nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization-based kinase in vitro assay using human PI3K alpha purchased from Echelon Biosciences and p110 alpha/p85 alpha from Upstate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University of Pennsylvania

LigandPNGBDBM36525(EAd125)
Affinity DataIC50:  180nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization-based kinase in vitro assay using human PI3K alpha purchased from Echelon Biosciences and p110 alpha/p85 alpha from Upstate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University of Pennsylvania

LigandPNGBDBM36524(DW12Me)
Affinity DataIC50:  500nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization-based kinase in vitro assay using human PI3K alpha purchased from Echelon Biosciences and p110 alpha/p85 alpha from Upstate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University of Pennsylvania

LigandPNGBDBM36525(EAd125)
Affinity DataIC50:  700nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization-based kinase in vitro assay using human PI3K alpha purchased from Echelon Biosciences and p110 alpha/p85 alpha from Upstate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University of Pennsylvania

LigandPNGBDBM36523(DW12)
Affinity DataIC50:  750nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization-based kinase in vitro assay using human PI3K alpha purchased from Echelon Biosciences and p110 alpha/p85 alpha from Upstate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University of Pennsylvania

LigandPNGBDBM36522(HB12)
Affinity DataIC50: >1.00E+3nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization-based kinase in vitro assay using human PI3K alpha purchased from Echelon Biosciences and p110 alpha/p85 alpha from Upstate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University of Pennsylvania

LigandPNGBDBM36524(DW12Me)
Affinity DataIC50: >1.00E+3nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization-based kinase in vitro assay using human PI3K alpha purchased from Echelon Biosciences and p110 alpha/p85 alpha from Upstate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University of Pennsylvania

LigandPNGBDBM36525(EAd125)
Affinity DataIC50:  4.00E+3nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization-based kinase in vitro assay using human PI3K alpha purchased from Echelon Biosciences and p110 alpha/p85 alpha from Upstate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed