Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50038497
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377205BDBM50377205(CHEMBL254582)
Affinity DataIC50: 200nMAssay Description:Inhibition of GSK3-beta by ATP-based competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377190BDBM50377190(CHEMBL427726)
Affinity DataIC50: 350nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377208BDBM50377208(CHEMBL402228)
Affinity DataIC50: 410nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377206BDBM50377206(CHEMBL253532)
Affinity DataIC50: 630nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377205BDBM50377205(CHEMBL254582)
Affinity DataIC50: 690nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377207BDBM50377207(CHEMBL257993)
Affinity DataIC50: 710nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377204BDBM50377204(CHEMBL257992)
Affinity DataIC50: 710nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377202BDBM50377202(CHEMBL254961)
Affinity DataIC50: 860nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377203BDBM50377203(CHEMBL403309)
Affinity DataIC50: 860nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377213BDBM50377213(CHEMBL401654)
Affinity DataIC50: 890nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377201BDBM50377201(CHEMBL254758)
Affinity DataIC50: 900nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377200BDBM50377200(CHEMBL255915)
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377192BDBM50377192(CHEMBL428252)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377199BDBM50377199(CHEMBL254794)
Affinity DataIC50: 1.33E+3nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377212BDBM50377212(CHEMBL255284)
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377198BDBM50377198(CHEMBL402325)
Affinity DataIC50: 1.48E+3nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377197BDBM50377197(CHEMBL402324)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377196BDBM50377196(CHEMBL258029)
Affinity DataIC50: 2.61E+3nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377211BDBM50377211(CHEMBL257823)
Affinity DataIC50: 2.99E+3nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377195BDBM50377195(CHEMBL403640)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377194BDBM50377194(CHEMBL256559)
Affinity DataIC50: 3.38E+3nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377210BDBM50377210(CHEMBL257980)
Affinity DataIC50: 3.48E+3nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377193BDBM50377193(CHEMBL257979)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377191BDBM50377191(CHEMBL256367)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377209BDBM50377209(CHEMBL257821)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of GSK3-beta assessed as breakdown of glycogen synthase derived substrate peptide by ADP hunter assay in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377208BDBM50377208(CHEMBL402228)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human recombinant Pim1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377190BDBM50377190(CHEMBL427726)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of GSK3-beta assessed as beta-casein level by RKO-cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377205BDBM50377205(CHEMBL254582)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of GSK3-beta assessed as beta-casein level by RKO-cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377207BDBM50377207(CHEMBL257993)
Affinity DataIC50: 1.92E+4nMAssay Description:Inhibition of GSK3-beta assessed as beta-casein level by RKO-cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377208BDBM50377208(CHEMBL402228)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of GSK3-beta assessed as beta-casein level by RKO-cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377192BDBM50377192(CHEMBL428252)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of GSK3-beta assessed as beta-casein level by RKO-cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed