Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50026229
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50176988(8-chloro-1-(2',4'-dichlorophenyl)-N-piperi...)
Affinity DataKi:  0.000350nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  1.18nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50176988(8-chloro-1-(2',4'-dichlorophenyl)-N-piperi...)
Affinity DataKi:  5.55nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50271287(5-(4-Chloro-2-methylphenyl)-1-(2,4-dichlorophenyl)...)
Affinity DataKi:  5.83nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  6.18nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50270540(9-Chloro-1-(2,4-dichlorophenyl)-N-piperidin-1-yl-4...)
Affinity DataKi:  14.7nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50176983(7-chloro-1-(2,4-dichlorophenyl)-N-(piperidin-1-yl)...)
Affinity DataKi:  15nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50271287(5-(4-Chloro-2-methylphenyl)-1-(2,4-dichlorophenyl)...)
Affinity DataKi:  16.1nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50271285(1,5-bis(2,4-Dichlorophenyl)-4-methyl-N-piperidin-1...)
Affinity DataKi:  17.9nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50176988(8-chloro-1-(2',4'-dichlorophenyl)-N-piperi...)
Affinity DataKi:  18.4nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50176988(8-chloro-1-(2',4'-dichlorophenyl)-N-piperi...)
Affinity DataKi:  20nMAssay Description:Binding affinity to CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50271285(1,5-bis(2,4-Dichlorophenyl)-4-methyl-N-piperidin-1...)
Affinity DataKi:  34.2nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50270540(9-Chloro-1-(2,4-dichlorophenyl)-N-piperidin-1-yl-4...)
Affinity DataKi:  40.9nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50270539(5-(4-Chloro-2,6-dimethylphenyl)-1-(2,4-dichlorophe...)
Affinity DataKi:  116nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50271286(5-(2,4-Dichlorophenyl)-4-methyl-N-piperidin-1-yl-1...)
Affinity DataKi:  148nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50271288(5-(4-Chloro-2-methylphenyl)-4-methyl-N-piperidin-1...)
Affinity DataKi:  152nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50270539(5-(4-Chloro-2,6-dimethylphenyl)-1-(2,4-dichlorophe...)
Affinity DataKi:  194nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50176983(7-chloro-1-(2,4-dichlorophenyl)-N-(piperidin-1-yl)...)
Affinity DataKi:  230nMAssay Description:Binding affinity to CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50271288(5-(4-Chloro-2-methylphenyl)-4-methyl-N-piperidin-1...)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50271286(5-(2,4-Dichlorophenyl)-4-methyl-N-piperidin-1-yl-1...)
Affinity DataKi:  261nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  313nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50270540(9-Chloro-1-(2,4-dichlorophenyl)-N-piperidin-1-yl-4...)
Affinity DataKi:  492nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50270539(5-(4-Chloro-2,6-dimethylphenyl)-1-(2,4-dichlorophe...)
Affinity DataKi:  758nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50271285(1,5-bis(2,4-Dichlorophenyl)-4-methyl-N-piperidin-1...)
Affinity DataKi:  1.04E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50271286(5-(2,4-Dichlorophenyl)-4-methyl-N-piperidin-1-yl-1...)
Affinity DataKi:  1.11E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50271287(5-(4-Chloro-2-methylphenyl)-1-(2,4-dichlorophenyl)...)
Affinity DataKi:  1.12E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50271288(5-(4-Chloro-2-methylphenyl)-4-methyl-N-piperidin-1...)
Affinity DataKi:  1.78E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed