Compile Data Set for Download or QSAR
maximum 50k data
Found 106 Enz. Inhib. hit(s) with all data for entry = 50026322
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243780(2-(dimethylamino)-1-(4-(6-phenyl-7-(4-((4-(5-(pyri...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(CHEMBL443661 | N,N-dimethyl-2-(4-(6-phenyl-7-(4-((...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Akt2 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(CHEMBL443661 | N,N-dimethyl-2-(4-(6-phenyl-7-(4-((...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243764(2-morpholino-6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4...)
Affinity DataIC50:  5nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243777(1-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4...)
Affinity DataIC50:  5nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243776(2-(1H-imidazol-1-yl)-6-phenyl-7-(4-((4-(5-(pyridin...)
Affinity DataIC50:  5nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24880(CHEMBL252857 | N-methyl-6-phenyl-7-[4-({4-[5-(pyri...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243780(2-(dimethylamino)-1-(4-(6-phenyl-7-(4-((4-(5-(pyri...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243783(2-(4-(1-methylazetidin-3-yl)piperazin-1-yl)-6-phen...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243780(2-(dimethylamino)-1-(4-(6-phenyl-7-(4-((4-(5-(pyri...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Akt2 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243765(1-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4-tr...)
Affinity DataIC50:  7nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243778(2-(4-(methylsulfonyl)piperazin-1-yl)-6-phenyl-7-(4...)
Affinity DataIC50:  7nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243769(2-((R)-3-methylpiperazin-1-yl)-6-phenyl-7-(4-((4-(...)
Affinity DataIC50:  8nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243771(2-(4-methylpiperazin-1-yl)-6-phenyl-7-(4-((4-(5-(p...)
Affinity DataIC50:  9nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243783(2-(4-(1-methylazetidin-3-yl)piperazin-1-yl)-6-phen...)
Affinity DataIC50:  9nMAssay Description:Inhibition of Akt2 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243782(2-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4...)
Affinity DataIC50:  9nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(CHEMBL443661 | N,N-dimethyl-2-(4-(6-phenyl-7-(4-((...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243775(CHEMBL454859 | N,N-dimethyl-1-(6-phenyl-7-(4-((4-(...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243783(2-(4-(1-methylazetidin-3-yl)piperazin-1-yl)-6-phen...)
Affinity DataIC50:  12nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243779(CHEMBL447348 | N,N-dimethyl-4-(6-phenyl-7-(4-((4-(...)
Affinity DataIC50:  13nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24867(1-(2-aminophenyl)-3-[({4-[2-(methylsulfanyl)-6-phe...)
Affinity DataIC50:  15nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243777(1-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4...)
Affinity DataIC50:  15nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243777(1-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4...)
Affinity DataIC50:  16nMAssay Description:Inhibition of Akt2 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243782(2-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4...)
Affinity DataIC50:  17nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243770(2-((S)-3-methylpiperazin-1-yl)-6-phenyl-7-(4-((4-(...)
Affinity DataIC50:  17nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243765(1-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4-tr...)
Affinity DataIC50:  17nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243779(CHEMBL447348 | N,N-dimethyl-4-(6-phenyl-7-(4-((4-(...)
Affinity DataIC50:  18nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243763(6-phenyl-2-(piperidin-1-yl)-7-(4-((4-(5-(pyridin-2...)
Affinity DataIC50:  18nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243780(2-(dimethylamino)-1-(4-(6-phenyl-7-(4-((4-(5-(pyri...)
Affinity DataIC50:  19nMAssay Description:Inhibition of Akt2 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243764(2-morpholino-6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4...)
Affinity DataIC50:  19nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243781(2-(5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)...)
Affinity DataIC50:  19nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243778(2-(4-(methylsulfonyl)piperazin-1-yl)-6-phenyl-7-(4...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243762(2-(3,3-difluoropyrrolidin-1-yl)-6-phenyl-7-(4-((4-...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24880(CHEMBL252857 | N-methyl-6-phenyl-7-[4-({4-[5-(pyri...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243775(CHEMBL454859 | N,N-dimethyl-1-(6-phenyl-7-(4-((4-(...)
Affinity DataIC50:  22nMAssay Description:Inhibition of Akt2 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243778(2-(4-(methylsulfonyl)piperazin-1-yl)-6-phenyl-7-(4...)
Affinity DataIC50:  23nMAssay Description:Inhibition of Akt2 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243775(CHEMBL454859 | N,N-dimethyl-1-(6-phenyl-7-(4-((4-(...)
Affinity DataIC50:  23nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243774((2R)-4-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2...)
Affinity DataIC50:  25nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243769(2-((R)-3-methylpiperazin-1-yl)-6-phenyl-7-(4-((4-(...)
Affinity DataIC50:  25nMAssay Description:Inhibition of Akt2 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243783(2-(4-(1-methylazetidin-3-yl)piperazin-1-yl)-6-phen...)
Affinity DataIC50:  27nMAssay Description:Inhibition of Akt2 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243771(2-(4-methylpiperazin-1-yl)-6-phenyl-7-(4-((4-(5-(p...)
Affinity DataIC50:  27nMAssay Description:Inhibition of Akt2 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243766(2-((2S,6R)-2,6-dimethylmorpholino)-6-phenyl-7-(4-(...)
Affinity DataIC50:  28nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243772(2-((2R,5S)-2,5-dimethylpiperazin-1-yl)-6-phenyl-7-...)
Affinity DataIC50:  29nMAssay Description:Inhibition of Akt2 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243782(2-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4...)
Affinity DataIC50:  31nMAssay Description:Inhibition of Akt2 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243776(2-(1H-imidazol-1-yl)-6-phenyl-7-(4-((4-(5-(pyridin...)
Affinity DataIC50:  35nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243769(2-((R)-3-methylpiperazin-1-yl)-6-phenyl-7-(4-((4-(...)
Affinity DataIC50:  36nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243771(2-(4-methylpiperazin-1-yl)-6-phenyl-7-(4-((4-(5-(p...)
Affinity DataIC50:  36nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243763(6-phenyl-2-(piperidin-1-yl)-7-(4-((4-(5-(pyridin-2...)
Affinity DataIC50:  36nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243767(2-(1,1-Dioxo-1lambda6-thiomorpholin-4-yl)-6-phenyl...)
Affinity DataIC50:  38nMAssay Description:Inhibition of Akt1 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(CHEMBL443661 | N,N-dimethyl-2-(4-(6-phenyl-7-(4-((...)
Affinity DataIC50:  39nMAssay Description:Inhibition of Akt2 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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