Compile Data Set for Download or QSAR
maximum 50k data
Found 48 Enz. Inhib. hit(s) with all data for entry = 50026392
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM85550(Ang IV | CAS_12676-15-2 | CHEMBL261120 | cid_12381...)
Affinity DataKi:  7nMAssay Description:Displacement of [125I]Angiotensin 4 from human recombinant IRAP expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM85550(Ang IV | CAS_12676-15-2 | CHEMBL261120 | cid_12381...)
Affinity DataKi:  60nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM85550(Ang IV | CAS_12676-15-2 | CHEMBL261120 | cid_12381...)
Affinity DataKi:  830nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242871(2-(2-(((2S,3R)-2-(3-(4-hydroxybenzyl)-5-((S)-2-ami...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [125I]Angiotensin 4 from human recombinant IRAP expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242861((S)-2-((S)-1-((S)-2-((2S,3S)-2-(3-(4-hydroxybenzyl...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242869(2-(2-(((2S,3R)-2-(3-(4-hydroxybenzyl)-5-((S)-2-ami...)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242868(2-(((2S,3R)-2-(3-(4-hydroxybenzyl)-5-((S)-2-amino-...)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242871(2-(2-(((2S,3R)-2-(3-(4-hydroxybenzyl)-5-((S)-2-ami...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242865(2-(2-(((S)-1-(3-(4-hydroxybenzyl)-5-((S)-2-aminohe...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [125I]Angiotensin 4 from human recombinant IRAP expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242870(2-(((2S,3R)-2-(3-(4-hydroxybenzyl)-5-((S)-2-aminoh...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242870(2-(((2S,3R)-2-(3-(4-hydroxybenzyl)-5-((S)-2-aminoh...)
Affinity DataKi:  2.30E+3nMAssay Description:Displacement of [125I]Angiotensin 4 from human recombinant IRAP expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242864(2-(((S)-1-(3-(4-hydroxybenzyl)-5-((S)-2-aminohexan...)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [125I]Angiotensin 4 from human recombinant IRAP expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242867(2-(2-(((S)-2-(3-(4-hydroxybenzyl)-5-((S)-2-aminohe...)
Affinity DataKi:  3.10E+3nMAssay Description:Displacement of [125I]Angiotensin 4 from human recombinant IRAP expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242865(2-(2-(((S)-1-(3-(4-hydroxybenzyl)-5-((S)-2-aminohe...)
Affinity DataKi:  3.30E+3nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242866(2-(((S)-2-(3-(4-hydroxybenzyl)-5-((S)-2-aminohexan...)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242866(2-(((S)-2-(3-(4-hydroxybenzyl)-5-((S)-2-aminohexan...)
Affinity DataKi:  3.90E+3nMAssay Description:Displacement of [125I]Angiotensin 4 from human recombinant IRAP expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242867(2-(2-(((S)-2-(3-(4-hydroxybenzyl)-5-((S)-2-aminohe...)
Affinity DataKi:  3.90E+3nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242861((S)-2-((S)-1-((S)-2-((2S,3S)-2-(3-(4-hydroxybenzyl...)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242864(2-(((S)-1-(3-(4-hydroxybenzyl)-5-((S)-2-aminohexan...)
Affinity DataKi:  6.30E+3nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242861((S)-2-((S)-1-((S)-2-((2S,3S)-2-(3-(4-hydroxybenzyl...)
Affinity DataKi:  6.80E+3nMAssay Description:Displacement of [125I]Angiotensin 4 from human recombinant IRAP expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242863(2-(2-(((S)-1-(3-(4-hydroxybenzyl)-5-((S)-2-amino-3...)
Affinity DataKi:  7.40E+3nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242869(2-(2-(((2S,3R)-2-(3-(4-hydroxybenzyl)-5-((S)-2-ami...)
Affinity DataKi:  8.90E+3nMAssay Description:Displacement of [125I]Angiotensin 4 from human recombinant IRAP expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242866(2-(((S)-2-(3-(4-hydroxybenzyl)-5-((S)-2-aminohexan...)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242865(2-(2-(((S)-1-(3-(4-hydroxybenzyl)-5-((S)-2-aminohe...)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242862(2-(((S)-1-(3-(4-hydroxybenzyl)-5-((S)-2-amino-3-me...)
Affinity DataKi:  1.20E+4nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242868(2-(((2S,3R)-2-(3-(4-hydroxybenzyl)-5-((S)-2-amino-...)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [125I]Angiotensin 4 from human recombinant IRAP expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242871(2-(2-(((2S,3R)-2-(3-(4-hydroxybenzyl)-5-((S)-2-ami...)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242862(2-(((S)-1-(3-(4-hydroxybenzyl)-5-((S)-2-amino-3-me...)
Affinity DataKi:  1.30E+4nMAssay Description:Displacement of [125I]Angiotensin 4 from human recombinant IRAP expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242863(2-(2-(((S)-1-(3-(4-hydroxybenzyl)-5-((S)-2-amino-3...)
Affinity DataKi:  1.40E+4nMAssay Description:Displacement of [125I]Angiotensin 4 from human recombinant IRAP expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242867(2-(2-(((S)-2-(3-(4-hydroxybenzyl)-5-((S)-2-aminohe...)
Affinity DataKi:  1.60E+4nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242938((S)-2-(2-((3-(4-hydroxybenzyl)-5-(2-amino-3-methyl...)
Affinity DataKi:  1.60E+4nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242864(2-(((S)-1-(3-(4-hydroxybenzyl)-5-((S)-2-aminohexan...)
Affinity DataKi:  1.70E+4nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242870(2-(((2S,3R)-2-(3-(4-hydroxybenzyl)-5-((S)-2-aminoh...)
Affinity DataKi:  1.70E+4nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242868(2-(((2S,3R)-2-(3-(4-hydroxybenzyl)-5-((S)-2-amino-...)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242869(2-(2-(((2S,3R)-2-(3-(4-hydroxybenzyl)-5-((S)-2-ami...)
Affinity DataKi:  2.10E+4nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242938((S)-2-(2-((3-(4-hydroxybenzyl)-5-(2-amino-3-methyl...)
Affinity DataKi:  3.30E+4nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50243085(2-(2-((3-(4-hydroxybenzyl)-5-aminobenzamido)methyl...)
Affinity DataKi:  3.50E+4nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242863(2-(2-(((S)-1-(3-(4-hydroxybenzyl)-5-((S)-2-amino-3...)
Affinity DataKi:  4.90E+4nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242862(2-(((S)-1-(3-(4-hydroxybenzyl)-5-((S)-2-amino-3-me...)
Affinity DataKi:  5.50E+4nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50243086((2S,3R)-2-(3-(4-hydroxybenzyl)-5-((S)-2-amino-3-me...)
Affinity DataKi:  6.90E+4nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50243086((2S,3R)-2-(3-(4-hydroxybenzyl)-5-((S)-2-amino-3-me...)
Affinity DataKi:  7.60E+4nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242938((S)-2-(2-((3-(4-hydroxybenzyl)-5-(2-amino-3-methyl...)
Affinity DataKi:  8.60E+4nMAssay Description:Displacement of [125I]Angiotensin 4 from human recombinant IRAP expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242872(2-(2-(((2S,3R)-2-(3-(4-hydroxybenzyl)-5-aminobenza...)
Affinity DataKi:  9.70E+4nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50243085(2-(2-((3-(4-hydroxybenzyl)-5-aminobenzamido)methyl...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50243086((2S,3R)-2-(3-(4-hydroxybenzyl)-5-((S)-2-amino-3-me...)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [125I]Angiotensin 4 from human recombinant IRAP expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50243085(2-(2-((3-(4-hydroxybenzyl)-5-aminobenzamido)methyl...)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [125I]Angiotensin 4 from human recombinant IRAP expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242872(2-(2-(((2S,3R)-2-(3-(4-hydroxybenzyl)-5-aminobenza...)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [125I]Angiotensin 4 from human recombinant IRAP expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50242872(2-(2-(((2S,3R)-2-(3-(4-hydroxybenzyl)-5-aminobenza...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed