Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 50038634
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50110288(CHEMBL15153 | N-(4-(3-(piperidin-1-yl)propoxy)phen...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]RAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50263054((6-(3-(piperidin-1-yl)propoxy)naphthalen-2-yl)(pyr...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]RAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50139391((R)-4-(2-(2-(2-methylpyrrolidin-1-yl)ethyl)benzofu...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]RAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50370569(A-349,821 | A-349821)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]RAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50263055((6-(1-isopropylpiperidin-4-yloxy)naphthalen-2-yl)(...)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]RAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50263096(CHEMBL477181 | N-cyclohexyl-6-(1-isopropylpiperidi...)
Affinity DataKi:  87nMAssay Description:Displacement of [3H]RAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50263096(CHEMBL477181 | N-cyclohexyl-6-(1-isopropylpiperidi...)
Affinity DataEC50:  21nMAssay Description:Inverse agonist activity at human histamine H3 receptor expressed in CHO cells by GTPgammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed