Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 50004066
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50183273BDBM50183273((S)-6-(3-chloro-2-fluorobenzyl)-1-(1-hydroxy-3-met...)
Affinity DataIC50: 2nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50183273BDBM50183273((S)-6-(3-chloro-2-fluorobenzyl)-1-(1-hydroxy-3-met...)
Affinity DataIC50: 7nMAssay Description:Inhibition of HIV1 integrase DNA strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50183276BDBM50183276(6-(3-chloro-2-fluorobenzyl)-1-(2-hydroxyethyl)-4-o...)
Affinity DataIC50: 24nMAssay Description:Inhibition of HIV1 integrase DNA strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479127BDBM50479127(CHEMBL522229)
Affinity DataIC50: 50nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50183273BDBM50183273((S)-6-(3-chloro-2-fluorobenzyl)-1-(1-hydroxy-3-met...)
Affinity DataIC50: 50nMAssay Description:Inhibition of HIV1 integrase 3'-processing activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479125BDBM50479125(CHEMBL458279)
Affinity DataIC50: 70nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479125BDBM50479125(CHEMBL458279)
Affinity DataIC50: 200nMAssay Description:Inhibition of HIV1 integrase DNA strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479127BDBM50479127(CHEMBL522229)
Affinity DataIC50: 600nMAssay Description:Inhibition of HIV1 integrase DNA strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479124BDBM50479124(CHEMBL458280)
Affinity DataIC50: 900nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479117BDBM50479117(CHEMBL497490)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479124BDBM50479124(CHEMBL458280)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of HIV1 integrase DNA strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479116BDBM50479116(CHEMBL497661)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of HIV1 integrase DNA strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479117BDBM50479117(CHEMBL497490)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of HIV1 integrase DNA strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479116BDBM50479116(CHEMBL497661)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479126BDBM50479126(CHEMBL511508)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479135BDBM50479135(CHEMBL526642)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479128BDBM50479128(CHEMBL497489)
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479134BDBM50479134(CHEMBL497505)
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479135BDBM50479135(CHEMBL526642)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of HIV1 integrase DNA strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479127BDBM50479127(CHEMBL522229)
Affinity DataIC50: 1.66E+4nMAssay Description:Inhibition of HIV1 integrase 3'-processing activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479126BDBM50479126(CHEMBL511508)
Affinity DataIC50: 1.85E+4nMAssay Description:Inhibition of HIV1 integrase DNA strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479123BDBM50479123(CHEMBL497506)
Affinity DataIC50: 1.87E+4nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479134BDBM50479134(CHEMBL497505)
Affinity DataIC50: 2.41E+4nMAssay Description:Inhibition of HIV1 integrase DNA strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479119BDBM50479119(CHEMBL498491)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479133BDBM50479133(CHEMBL498504)
Affinity DataIC50: 4.37E+4nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479131BDBM50479131(CHEMBL496491)
Affinity DataIC50: 5.49E+4nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479133BDBM50479133(CHEMBL498504)
Affinity DataIC50: 5.87E+4nMAssay Description:Inhibition of HIV1 integrase DNA strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479121BDBM50479121(CHEMBL497475)
Affinity DataIC50: 7.19E+4nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479122BDBM50479122(CHEMBL496476)
Affinity DataIC50: 7.39E+4nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479118BDBM50479118(CHEMBL526269)
Affinity DataIC50: 7.76E+4nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479115BDBM50479115(CHEMBL458483)
Affinity DataIC50: 8.69E+4nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479129BDBM50479129(CHEMBL444410)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479123BDBM50479123(CHEMBL497506)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 integrase 3'-processing activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479130BDBM50479130(CHEMBL498490)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 integrase DNA strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479120BDBM50479120(CHEMBL497476)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 integrase DNA strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479131BDBM50479131(CHEMBL496491)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 integrase DNA strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479121BDBM50479121(CHEMBL497475)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 integrase DNA strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479128BDBM50479128(CHEMBL497489)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 integrase DNA strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479129BDBM50479129(CHEMBL444410)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 integrase DNA strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479130BDBM50479130(CHEMBL498490)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479119BDBM50479119(CHEMBL498491)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 integrase DNA strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479122BDBM50479122(CHEMBL496476)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 integrase 3'-processing activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479123BDBM50479123(CHEMBL497506)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 integrase DNA strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479132BDBM50479132(CHEMBL498321)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479115BDBM50479115(CHEMBL458483)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 integrase DNA strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479119BDBM50479119(CHEMBL498491)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 integrase 3'-processing activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479131BDBM50479131(CHEMBL496491)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 integrase 3'-processing activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479118BDBM50479118(CHEMBL526269)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 integrase 3'-processing activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479120BDBM50479120(CHEMBL497476)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 integrase by overall integration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50479128BDBM50479128(CHEMBL497489)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 integrase 3'-processing activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
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