Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50048862
TargetType-1/Type-2 angiotensin II receptor(Human)
Berlex Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229504BDBM50229504(Saralasin)
Affinity DataIC50: 0.0660nMAssay Description:Inhibitory activity as antagonist of AII on guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Berlex Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030815BDBM50030815(CHEMBL404594)
Affinity DataIC50: 0.210nMAssay Description:Inhibitory activity as antagonist of AII on guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Berlex Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229420BDBM50229420(CHEMBL77838)
Affinity DataIC50: 0.450nMAssay Description:Inhibitory activity as antagonist of AII on guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Berlex Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50228894BDBM50228894(CHEMBL312754)
Affinity DataIC50: 5.80nMAssay Description:Inhibitory activity as antagonist of AII on guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Berlex Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229419BDBM50229419(CHEMBL405381)
Affinity DataIC50: 7nMAssay Description:The compound was tested for its ability to displace [3H]Angiotensin II (300 ng/mL) from rabbit adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Berlex Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229417BDBM50229417(CHEMBL2369863)
Affinity DataIC50: 330nMAssay Description:Inhibitory activity as antagonist of AII on guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Berlex Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229502BDBM50229502(CHEMBL308824)
Affinity DataIC50: 1.50E+4nMAssay Description:The compound was tested for its inhibitory activity as antagonist of AII on guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Berlex Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229418BDBM50229418(CHEMBL76890)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity as antagonist of AII on guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Berlex Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229503BDBM50229503(CHEMBL309651)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity as antagonist of AII on guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Berlex Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229421BDBM50229421(CHEMBL418901)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity as antagonist of AII on guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2019
Entry Details Article
PubMed