Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50000758
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM50009591(cis-1-(2-Methyl-1-phenyl-cyclohexyl)-piperidine | ...)
Affinity DataKi:  11nMAssay Description:Binding affinity by displacement of [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate preparation of rat brain without ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM50009591(cis-1-(2-Methyl-1-phenyl-cyclohexyl)-piperidine | ...)
Affinity DataKi:  25nMAssay Description:Binding affinity by displacement of [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate preparation of rat brain without ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM83449(cid_9795678 | PHENCYCLIDINE | SMR001338811 | Phenc...)
Affinity DataKi:  53nMAssay Description:Binding affinity by displacement of [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate preparation of rat brain without ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM50009592(CHEMBL424610 | cis-1-(4-Methyl-1-phenyl-cyclohexyl...)
Affinity DataKi:  617nMAssay Description:Binding affinity by displacement of [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate preparation of rat brain without ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM50009592(CHEMBL424610 | cis-1-(4-Methyl-1-phenyl-cyclohexyl...)
Affinity DataKi:  617nMAssay Description:Binding affinity by displacement of [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate preparation of rat brain without ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM50009591(cis-1-(2-Methyl-1-phenyl-cyclohexyl)-piperidine | ...)
Affinity DataKi:  2.18E+3nMAssay Description:Binding affinity by displacement of [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate preparation of rat brain without ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM50009591(cis-1-(2-Methyl-1-phenyl-cyclohexyl)-piperidine | ...)
Affinity DataKi:  2.94E+3nMAssay Description:Binding affinity by displacement of [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate preparation of rat brain without ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM50009590(CHEMBL86824 | cis-C-(2-Methyl-1-piperidin-1-yl-cyc...)
Affinity DataKi:  4.70E+3nMAssay Description:Binding affinity by displacement of [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate preparation of rat brain without ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM50009590(CHEMBL86824 | cis-C-(2-Methyl-1-piperidin-1-yl-cyc...)
Affinity DataKi:  4.70E+3nMAssay Description:Binding affinity by displacement of [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate preparation of rat brain without ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM50009591(cis-1-(2-Methyl-1-phenyl-cyclohexyl)-piperidine | ...)
Affinity DataKi:  7.40E+3nMAssay Description:Binding affinity by displacement of [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate preparation of rat brain without ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM50009591(cis-1-(2-Methyl-1-phenyl-cyclohexyl)-piperidine | ...)
Affinity DataKi:  7.40E+3nMAssay Description:Binding affinity by displacement of [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate preparation of rat brain without ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM50009593(CHEMBL89477 | C-Phenyl-C-(1-piperidin-1-yl-cyclohe...)
Affinity DataKi:  3.10E+4nMAssay Description:Binding affinity by displacement of [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate preparation of rat brain without ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed