Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50027122
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8611BDBM8611(CHEMBL468419 | 4-{5H,6H,7H,8H-imidazo[1,5-a]pyridi...)
Affinity DataIC50: 50nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263871BDBM50263871(1-[2-Biphenyl-4-yl-1-(4-fluoro-benzyl)-ethyl]-1H-i...)
Affinity DataIC50: 110nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263761BDBM50263761(Biphenyl-4-ylmethyl-(4-fluoro-benzyl)-imidazol-1-y...)
Affinity DataIC50: 190nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263924BDBM50263924(1-[2-Biphenyl-4-yl-1-(2,4-difluoro-benzyl)-ethyl]-...)
Affinity DataIC50: 260nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263719BDBM50263719(Biphenyl-4-ylmethyl-(2-chloro-benzyl)-imidazol-1-y...)
Affinity DataIC50: 300nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263461BDBM50263461(N-(5-chlorothiophen-2-ylmethyl)-N-(2,4-dichloroben...)
Affinity DataIC50: 320nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263808BDBM50263808(Biphenyl-4-ylmethyl-(2,4-difluoro-benzyl)-imidazol...)
Affinity DataIC50: 350nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263720BDBM50263720(Biphenyl-4-ylmethyl-(2-fluoro-benzyl)-imidazol-1-y...)
Affinity DataIC50: 460nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263921BDBM50263921(1-[2-Biphenyl-4-yl-1-(2-methoxy-benzyl)-ethyl]-1H-...)
Affinity DataIC50: 510nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263810BDBM50263810(N-(4-tert-butylbenzyl)-N-(thiophen-2-ylmethyl)-1H-...)
Affinity DataIC50: 580nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263465BDBM50263465(1-(5-chlorothiophen-2-yl)-2-(1H-imidazol-1-yl)-3-p...)
Affinity DataIC50: 870nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263812BDBM50263812(1-(1-Benzyl-2-biphenyl-4-yl-ethyl)-1H-imidazole | ...)
Affinity DataIC50: 950nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263811BDBM50263811(1-[2-Biphenyl-4-yl-1-(4-tert-butyl-benzyl)-ethyl]-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263867BDBM50263867(1-[2-Biphenyl-4-yl-1-(2-methyl-benzyl)-ethyl]-1H-i...)
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263343BDBM50263343(N-(1,1'-biphenyl-4-ylmethyl)-N-(5-chlorothiophen-2...)
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263368BDBM50263368(N-benzyl-N-(5-chlorothiophen-2-yl-methyl)-1H-imida...)
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263464BDBM50263464(1-(1,1'-biphenyl-4-yl)-3-(5-chloro-thiophen-2-yl)-...)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263868BDBM50263868(1-[2-Biphenyl-4-yl-1-(2-chloro-benzyl)-ethyl]-1H-i...)
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263760BDBM50263760(Biphenyl-4-ylmethyl-(4-chloro-benzyl)-imidazol-1-y...)
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263717BDBM50263717(Benzyl-biphenyl-4-ylmethyl-imidazol-1-yl-amine | C...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263923BDBM50263923(1-[2-Biphenyl-4-yl-1-(2,4-dichloro-benzyl)-ethyl]-...)
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263870BDBM50263870(1-[2-Biphenyl-4-yl-1-(4-methyl-benzyl)-ethyl]-1H-i...)
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263869BDBM50263869(1-[2-Biphenyl-4-yl-1-(2-fluoro-benzyl)-ethyl]-1H-i...)
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263762BDBM50263762(Biphenyl-4-ylmethyl-imidazol-1-yl-(2-methoxy-benzy...)
Affinity DataIC50: 1.51E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263809BDBM50263809(N-(2,4-dichlorobenzyl)-N-(4-tert-butylbenzyl)-1H-i...)
Affinity DataIC50: 1.52E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263763BDBM50263763(Biphenyl-4-ylmethyl-imidazol-1-yl-(4-methoxy-benzy...)
Affinity DataIC50: 1.53E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263922BDBM50263922(1-[2-Biphenyl-4-yl-1-(4-methoxy-benzyl)-ethyl]-1H-...)
Affinity DataIC50: 1.68E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263666BDBM50263666(Biphenyl-4-ylmethyl-(4-tert-butyl-benzyl)-imidazol...)
Affinity DataIC50: 2.16E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263721BDBM50263721(Biphenyl-4-ylmethyl-imidazol-1-yl-(4-methyl-benzyl...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263463BDBM50263463(N-(benzo[b]thiophen-7-ylmethyl)-N-(2,4-dichloroben...)
Affinity DataIC50: 2.49E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263718BDBM50263718(Biphenyl-4-ylmethyl-imidazol-1-yl-(2-methyl-benzyl...)
Affinity DataIC50: 2.96E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263764BDBM50263764(Biphenyl-4-ylmethyl-(2,4-dichloro-benzyl)-imidazol...)
Affinity DataIC50: 3.65E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263665BDBM50263665(N-(2,4-dichlorobenzyl)-N-(naphthalen-1-ylmethyl)-1...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263664BDBM50263664(N-(4-tert-butylbenzyl)-N-(naphthalen-1-ylmethyl)-1...)
Affinity DataIC50: 4.59E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263341BDBM50263341(N-(4-tert-butylbenzyl)-N-(4-phenylbut-3-enyl)-1H-1...)
Affinity DataIC50: 5.06E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263342BDBM50263342(N-(4-tert-butylbenzyl)-N-(thiophen-2-ylmethyl)-1H-...)
Affinity DataIC50: 9.23E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263462BDBM50263462(N-benzyl-N-(benzo[b]thiophen-7-ylmethyl)-1H-imidaz...)
Affinity DataIC50: 9.96E+3nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50264032BDBM50264032(N-(naphthalen-1-ylmethyl)-N-(4-phenylbut-3-enyl)-1...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAromatase(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50263340BDBM50263340(N-(2,4-dichlorobenzyl)-N-(4-phenylbut-3-enyl)-1H-1...)
Affinity DataIC50: 1.73E+4nMAssay Description:Inhibition of human aromataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed