Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50027217
TargetAlpha-2A adrenergic receptor(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50253285(4-Bromo-N-(3-bromo-4-(3-(dimethylamino)propoxy)phe...)
Affinity DataKi:  69nMAssay Description:Displacement of [3H]MK912 from human cloned adrenergic alpha-2a receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50253285(4-Bromo-N-(3-bromo-4-(3-(dimethylamino)propoxy)phe...)
Affinity DataIC50: 185nMAssay Description:Displacement of [3H]MK912 from human cloned adrenergic alpha-2a receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50253285(4-Bromo-N-(3-bromo-4-(3-(dimethylamino)propoxy)phe...)
Affinity DataKi:  275nMAssay Description:Inhibition of cloned adrenergic Alpha-1D receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50253285(4-Bromo-N-(3-bromo-4-(3-(dimethylamino)propoxy)phe...)
Affinity DataIC50: 560nMAssay Description:Inhibition of cloned adrenergic Alpha-1D receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50253285(4-Bromo-N-(3-bromo-4-(3-(dimethylamino)propoxy)phe...)
Affinity DataKi:  1.02E+3nMAssay Description:Displacement of [125I]-APT from histamine H2 receptor in brain of guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50253285(4-Bromo-N-(3-bromo-4-(3-(dimethylamino)propoxy)phe...)
Affinity DataKi:  1.04E+3nMAssay Description:Displacement of [3H]SMT from histamine H3 receptor in forebrain of ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50253285(4-Bromo-N-(3-bromo-4-(3-(dimethylamino)propoxy)phe...)
Affinity DataIC50: 1.25E+3nMAssay Description:Displacement of [125I]-APT from histamine H2 receptor in brain of guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50253285(4-Bromo-N-(3-bromo-4-(3-(dimethylamino)propoxy)phe...)
Affinity DataIC50: 2.35E+3nMAssay Description:Displacement of [3H]SMT from histamine H3 receptor in forebrain of ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed