Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50038767
TargetRyanodine receptor 1(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50191286BDBM50191286(Bastadin-5 | bastadin 5 | CHEMBL439151)
Affinity DataEC50:  2.20E+3nMAssay Description:Binding affinity to RYR1 channels by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetRyanodine receptor 1(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50191280BDBM50191280(5,21-Dibromo-4-hydroxy-2-oxa-10,14-diaza-tricyclo[...)
Affinity DataIC50: 6.00E+3nMAssay Description:Binding affinity to RYR1 channels by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetRyanodine receptor 1(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50150778BDBM50150778(polybrominated diphenyl ether derivative | Bastadi...)
Affinity DataEC50:  6.30E+3nMAssay Description:Binding affinity to RYR1 channels by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetRyanodine receptor 1(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50191278BDBM50191278((+/-)-5,17-dibromo-4-hydroxy-2-oxa-10-aza-tricyclo...)
Affinity DataEC50:  1.10E+4nMAssay Description:Binding affinity to RYR1 channels by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetRyanodine receptor 1(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50241985BDBM50241985(CHEMBL508830 | Bastadin-19 | CHEMBL506286 | (E,Z)b...)
Affinity DataEC50: >1.00E+5nMAssay Description:Binding affinity to RYR1 channels by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed