Compile Data Set for Download or QSAR
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Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50038767
TargetRyanodine receptor 1(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50191280(5,21-Dibromo-4-hydroxy-2-oxa-10,14-diaza-tricyclo[...)
Affinity DataIC50:  6.00E+3nMAssay Description:Binding affinity to RYR1 channels by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRyanodine receptor 1(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50241985((E,Z)bastadin-19 | Bastadin-19 | CHEMBL506286 | CH...)
Affinity DataEC50: >1.00E+5nMAssay Description:Binding affinity to RYR1 channels by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRyanodine receptor 1(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50150778(Bastadin-7 | Bastadins 7 | CHEMBL360190 | bastadin...)
Affinity DataEC50:  6.30E+3nMAssay Description:Binding affinity to RYR1 channels by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRyanodine receptor 1(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50191278((+/-)-5,17-dibromo-4-hydroxy-2-oxa-10-aza-tricyclo...)
Affinity DataEC50:  1.10E+4nMAssay Description:Binding affinity to RYR1 channels by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRyanodine receptor 1(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50191286(Bastadin-5 | CHEMBL439151 | bastadin 5)
Affinity DataEC50:  2.20E+3nMAssay Description:Binding affinity to RYR1 channels by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed