Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with all data for entry = 2965
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26429BDBM26429(CHEMBL511829 | (2E)-3-{4-[({8-carbamoyl-7-[(3,5-di...)
Affinity DataIC50: 47nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26428BDBM26428(ethyl (2E)-3-{4-[({8-carbamoyl-7-[(3,5-dimethoxyph...)
Affinity DataIC50: 88nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26415BDBM26415(5-{[(2,4-difluorophenyl)methyl]amino}-7-[(3,5-dime...)
Affinity DataIC50: 150nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26419BDBM26419(7-[(3,5-dimethoxyphenyl)amino]-5-{[(4-sulfamoylphe...)
Affinity DataIC50: 150nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26422BDBM26422(4-[({8-carbamoyl-7-[(3,5-dimethoxyphenyl)amino]imi...)
Affinity DataIC50: 180nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26420BDBM26420(7-[(3,5-dimethoxyphenyl)amino]-5-{[(4-methanesulfo...)
Affinity DataIC50: 190nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26418BDBM26418(5-[(1H-1,3-benzodiazol-2-ylmethyl)amino]-7-[(3,5-d...)
Affinity DataIC50: 200nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26410BDBM26410(7-[(3,5-dimethoxyphenyl)amino]-5-{[(4-fluorophenyl...)
Affinity DataIC50: 220nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26404BDBM26404(5-[(2-aminoethyl)amino]-7-[(3,5-dimethoxyphenyl)am...)
Affinity DataIC50: 230nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26411BDBM26411(7-[(3,5-dimethoxyphenyl)amino]-5-{[(4-methoxypheny...)
Affinity DataIC50: 230nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26426BDBM26426(2-{4-[({8-carbamoyl-7-[(3,5-dimethoxyphenyl)amino]...)
Affinity DataIC50: 240nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26416BDBM26416(7-[(3,5-dimethoxyphenyl)amino]-5-[(pyridin-4-ylmet...)
Affinity DataIC50: 250nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26413BDBM26413(7-[(3,5-dimethoxyphenyl)amino]-5-{[(2-methoxypheny...)
Affinity DataIC50: 340nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26405BDBM26405(5-(benzylamino)-7-[(3,5-dimethoxyphenyl)amino]imid...)
Affinity DataIC50: 400nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26408BDBM26408(7-[(3,5-dimethoxyphenyl)amino]-5-{[(1R)-1-phenylet...)
Affinity DataIC50: 410nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26421BDBM26421(methyl 4-[({8-carbamoyl-7-[(3,5-dimethoxyphenyl)am...)
Affinity DataIC50: 420nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26427BDBM26427(5-({[4-(carbamoylmethyl)phenyl]methyl}amino)-7-[(3...)
Affinity DataIC50: 480nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26412BDBM26412(7-[(3,5-dimethoxyphenyl)amino]-5-{[(3-methoxypheny...)
Affinity DataIC50: 530nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26423BDBM26423(5-{[(4-carbamoylphenyl)methyl]amino}-7-[(3,5-dimet...)
Affinity DataIC50: 660nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26424BDBM26424(7-[(3,5-dimethoxyphenyl)amino]-5-({[4-(hydroxymeth...)
Affinity DataIC50: 690nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26429BDBM26429(CHEMBL511829 | (2E)-3-{4-[({8-carbamoyl-7-[(3,5-di...)
Affinity DataIC50: 690nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26426BDBM26426(2-{4-[({8-carbamoyl-7-[(3,5-dimethoxyphenyl)amino]...)
Affinity DataIC50: 760nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26414BDBM26414(5-{[(3,5-difluorophenyl)methyl]amino}-7-[(3,5-dime...)
Affinity DataIC50: 910nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26417BDBM26417(7-[(3,5-dimethoxyphenyl)amino]-5-[(furan-2-ylmethy...)
Affinity DataIC50: 920nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26409BDBM26409(7-[(3,5-dimethoxyphenyl)amino]-5-{[(1S)-1-phenylet...)
Affinity DataIC50: 930nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26403BDBM26403(7-[(3,5-dimethoxyphenyl)amino]-5-[(2-hydroxyethyl)...)
Affinity DataIC50: 1.90E+3nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26410BDBM26410(7-[(3,5-dimethoxyphenyl)amino]-5-{[(4-fluorophenyl...)
Affinity DataIC50: 1.90E+3nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26427BDBM26427(5-({[4-(carbamoylmethyl)phenyl]methyl}amino)-7-[(3...)
Affinity DataIC50: 1.90E+3nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26416BDBM26416(7-[(3,5-dimethoxyphenyl)amino]-5-[(pyridin-4-ylmet...)
Affinity DataIC50: 2.30E+3nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26417BDBM26417(7-[(3,5-dimethoxyphenyl)amino]-5-[(furan-2-ylmethy...)
Affinity DataIC50: 2.50E+3nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26401BDBM26401(7-[(3,5-dimethoxyphenyl)amino]-5-(methylsulfanyl)i...)
Affinity DataIC50: 3.00E+3nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26425BDBM26425(tert-butyl 2-{4-[({8-carbamoyl-7-[(3,5-dimethoxyph...)
Affinity DataIC50: 3.20E+3nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26409BDBM26409(7-[(3,5-dimethoxyphenyl)amino]-5-{[(1S)-1-phenylet...)
Affinity DataIC50: 3.30E+3nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26404BDBM26404(5-[(2-aminoethyl)amino]-7-[(3,5-dimethoxyphenyl)am...)
Affinity DataIC50: 3.50E+3nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26415BDBM26415(5-{[(2,4-difluorophenyl)methyl]amino}-7-[(3,5-dime...)
Affinity DataIC50: 3.70E+3nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26403BDBM26403(7-[(3,5-dimethoxyphenyl)amino]-5-[(2-hydroxyethyl)...)
Affinity DataIC50: 4.30E+3nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26405BDBM26405(5-(benzylamino)-7-[(3,5-dimethoxyphenyl)amino]imid...)
Affinity DataIC50: 4.30E+3nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26421BDBM26421(methyl 4-[({8-carbamoyl-7-[(3,5-dimethoxyphenyl)am...)
Affinity DataIC50: 4.80E+3nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26407BDBM26407(7-[(3,5-dimethoxyphenyl)amino]-5-[(2-phenylethyl)a...)
Affinity DataIC50: 4.80E+3nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26407BDBM26407(7-[(3,5-dimethoxyphenyl)amino]-5-[(2-phenylethyl)a...)
Affinity DataIC50: 5.10E+3nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26406BDBM26406(5-[benzyl(methyl)amino]-7-[(3,5-dimethoxyphenyl)am...)
Affinity DataIC50: 5.50E+3nMpH: 7.6 T: 2°CAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26413BDBM26413(7-[(3,5-dimethoxyphenyl)amino]-5-{[(2-methoxypheny...)
Affinity DataIC50: 5.80E+3nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26412BDBM26412(7-[(3,5-dimethoxyphenyl)amino]-5-{[(3-methoxypheny...)
Affinity DataIC50: 6.70E+3nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26402BDBM26402(5-amino-7-[(3,5-dimethoxyphenyl)amino]imidazo[1,2-...)
Affinity DataIC50: 7.10E+3nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26422BDBM26422(4-[({8-carbamoyl-7-[(3,5-dimethoxyphenyl)amino]imi...)
Affinity DataIC50: 8.10E+3nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26424BDBM26424(7-[(3,5-dimethoxyphenyl)amino]-5-({[4-(hydroxymeth...)
Affinity DataIC50: 8.50E+3nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26423BDBM26423(5-{[(4-carbamoylphenyl)methyl]amino}-7-[(3,5-dimet...)
Affinity DataIC50: 8.70E+3nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26418BDBM26418(5-[(1H-1,3-benzodiazol-2-ylmethyl)amino]-7-[(3,5-d...)
Affinity DataIC50: 9.80E+3nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26414BDBM26414(5-{[(3,5-difluorophenyl)methyl]amino}-7-[(3,5-dime...)
Affinity DataIC50: 9.80E+3nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Kissei Pharmaceutical

LigandChemical structure of BindingDB Monomer ID 26401BDBM26401(7-[(3,5-dimethoxyphenyl)amino]-5-(methylsulfanyl)i...)
Affinity DataIC50: 1.00E+4nMAssay Description:A coupled spectrophotometric assay was used wherein ADP generated by ZAP-70 kinase was converted to ATP by pyruvate kinase (PK), with concomitant pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2009
Entry Details Article
PubMed
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