Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50027744
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50265823(CHEMBL516634 | candelalide B)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of voltage-gated Kv1.3 potassium channel (unknown origin) expressed in CHO cells by 86Rb efflux experimentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50265824(CHEMBL460814 | candelalide C)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of voltage-gated Kv1.3 potassium channel (unknown origin) expressed in CHO cells by 86Rb efflux experimentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50266317(CHEMBL515037 | candelalide A)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of voltage-gated Kv1.3 potassium channel (unknown origin) expressed in CHO cells by 86Rb efflux experimentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50265825(CHEMBL516932 | Nalanthalide)
Affinity DataIC50:  3.90E+3nMAssay Description:Antagonist activity at voltage-gated Kv1.3 potassium channel (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed