Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50030263
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50279106BDBM50279106(5-(4-phenoxybutoxy)psoralen | 4-(4-phenoxybutoxy)-...)
Affinity DataIC50: 2nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293351BDBM50293351(4-(4-Phenoxybutoxy)-7H-furo[3,2-g]chromene-7-thion...)
Affinity DataIC50: 17nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293343BDBM50293343(5-(4-Phenoxybutoxy)-2H-[1]benzopyran-2-one | CHEMB...)
Affinity DataIC50: 150nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293338BDBM50293338(6,7-Dimethoxy-4-(4-phenoxybutoxy)furo[2,3-b]quinol...)
Affinity DataIC50: 150nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293337BDBM50293337(9,10-Dihydro-4-methoxy-N-(4-phenoxybutyl)acridin-9...)
Affinity DataIC50: 165nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293345BDBM50293345(4-(4-Phenoxybutoxy)-5H-furo[3,2-g][1]benzopyran-5-...)
Affinity DataIC50: 170nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293339BDBM50293339(7,8-Dimethoxy-4-(4-phenoxybutoxy)furo[2,3-b]quinol...)
Affinity DataIC50: 200nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293340BDBM50293340(7-Methyl-4-(4-phenoxybutoxy)-5H-furo[3,2-g][1]benz...)
Affinity DataIC50: 233nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293348BDBM50293348(5-Methoxy-4-methyl-8-(4-phenoxybutoxy)psoralen | C...)
Affinity DataIC50: 318nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293334BDBM50293334(5,8-Dimethoxy-4-(4-phenoxybutoxy)psoralen | CHEMBL...)
Affinity DataIC50: 450nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293330BDBM50293330(5-(4-Phenoxybutoxy)isoquinoline | CHEMBL549464)
Affinity DataIC50: 520nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293344BDBM50293344(4-(4-Phenoxybutoxy)benzofuran | CHEMBL559956)
Affinity DataIC50: 650nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293331BDBM50293331(1,2-Dihydro-N-methyl-4-(4-phenoxybutoxy)quinolin-2...)
Affinity DataIC50: 670nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293332BDBM50293332(4-(4-Phenoxybutoxy)-2H-[1]benzopyran-2-one | CHEMB...)
Affinity DataIC50: 890nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293333BDBM50293333(3-(4-Phenoxybutoxy)-2-phenyl-4H-[1]benzopyran-4-on...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293349BDBM50293349(4-(4-Phenoxybutoxy)furo[2,3-b]quinoline | CHEMBL55...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293350BDBM50293350(9-(4-Phenoxybutyl)furo[2,3-b]quinolin-4(9H)-one | ...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293342BDBM50293342(8-(4-Phenoxybutoxy)psoralen | CHEMBL551028)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293341BDBM50293341(9-Methoxy-7-methyl-4-(4-phenoxybutoxy)-5H-furo[3,2...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293346BDBM50293346(2-Methyl-6,7-methylenedioxy-5-(4-phenoxybutoxy)-4H...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293347BDBM50293347(2,6-Dihydro-8-methyl-5-(4-phenoxybutoxy)pyrano[3,2...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293336BDBM50293336(1-(4-Phenoxybutoxy)anthraquinone | CHEMBL549316)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293329BDBM50293329(4-(4-Phenoxybutoxy)quinoline | CHEMBL564031)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293335BDBM50293335(9-(Phenoxybutoxy)-9H-dibenzo[b,e]pyran | CHEMBL550...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293328BDBM50293328(1-(4-Phenoxybutoxy)naphthalene | CHEMBL539158)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293327BDBM50293327(1,1'[1,4-Butanediyl(oxy)]bis-benzene | CHEMBL56254...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50067880BDBM50067880(4-methoxy-7H-furo[3,2-g]chromen-7-one | 5-methoxyp...)
Affinity DataIC50: 1.01E+5nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed