Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50027858
TargetTranscription factor Jun(Human)
B.V. Patel Pharmaceutical Education and Research Development Centre

Curated by ChEMBL
LigandPNGBDBM50279431(3-(4-Chloro-phenyl)-2-[2-(4-chloro-phenylamino)-4-...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of AP1 expressed in HEK293 cells assessed as inhibition of TNF-alpha-induced transcriptional activation treated 24 hrs before TNFalpha cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
B.V. Patel Pharmaceutical Education and Research Development Centre

Curated by ChEMBL
LigandPNGBDBM50279429(3-(4-Chloro-phenyl)-2-(4-methyl-2-methylamino-thia...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of AP1 expressed in HEK293 cells assessed as inhibition of TNF-alpha-induced transcriptional activation treated 24 hrs before TNFalpha cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
B.V. Patel Pharmaceutical Education and Research Development Centre

Curated by ChEMBL
LigandPNGBDBM50279699(2-(4-Methyl-2-phenylamino-thiazol-5-yl)-3-o-tolyl-...)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of AP1 expressed in HEK293 cells assessed as inhibition of TNF-alpha-induced transcriptional activation treated 24 hrs before TNFalpha cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
B.V. Patel Pharmaceutical Education and Research Development Centre

Curated by ChEMBL
LigandPNGBDBM50279698(2-(4-Methyl-2-methylamino-thiazol-5-yl)-3-o-tolyl-...)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of AP1 expressed in HEK293 cells assessed as inhibition of TNF-alpha-induced transcriptional activation treated 24 hrs before TNFalpha cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed