Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50027977
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179883BDBM50179883((4-Isopropylphenyl)-(4-isoquinolin-5-yl-phthalazin...)
Affinity DataIC50: 17nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21BDBM21(VANDETANIB | N-(4-bromo-2-fluorophenyl)-6-methoxy-...)
Affinity DataIC50: 45nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179881BDBM50179881(IM-094882 | N-(4-chlorophenyl)-4-(isoquinolin-5-yl...)
Affinity DataIC50: 48nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179890BDBM50179890((4-tert-Butylphenyl)-(4-isoquinolin-5-yl-phthalazi...)
Affinity DataIC50: 75nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173019BDBM50173019(4-[4-(4-tert-Butyl-phenylamino)-phthalazin-1-yl]-b...)
Affinity DataIC50: 78nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179889BDBM50179889([4-(Chloro-difluoro-methoxy)-phenyl]-(4-isoquinoli...)
Affinity DataIC50: 79nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173031BDBM50173031(4-(4-(4-bromophenylamino)phthalazin-1-yl)benzamide...)
Affinity DataIC50: 100nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179888BDBM50179888(N-(3,4-dichlorophenyl)-4-(isoquinolin-5-yl)phthala...)
Affinity DataIC50: 110nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179891BDBM50179891(N-(4-chloro-3-(trifluoromethyl)phenyl)-4-(isoquino...)
Affinity DataIC50: 120nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173045BDBM50173045(4-(4-(4-tert-butylphenylamino)phthalazin-1-yl)-N-m...)
Affinity DataIC50: 130nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173049BDBM50173049(4-{4-[4-(Chloro-difluoro-methoxy)-phenylamino]-pht...)
Affinity DataIC50: 190nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179893BDBM50179893(4-(isoquinolin-5-yl)-N-(2-methyl-1H-indol-5-yl)pht...)
Affinity DataIC50: 230nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179884BDBM50179884((4-Isoquinolin-5-yl-phthalazin-1-yl)-m-tolylamine ...)
Affinity DataIC50: 270nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179894BDBM50179894(4-(isoquinolin-5-yl)-N-(4-morpholinophenyl)phthala...)
Affinity DataIC50: 390nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173022BDBM50173022(3-[4-(4-tert-Butyl-phenylamino)-phthalazin-1-yl]-b...)
Affinity DataIC50: 400nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179882BDBM50179882((2-Fluoro-4-methylphenyl)-(4-isoquinolin-5-ylphtha...)
Affinity DataIC50: 430nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173034BDBM50173034(4-(4-(3-tert-butylphenylamino)phthalazin-1-yl)benz...)
Affinity DataIC50: 470nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173021BDBM50173021(4-{4-[4-(Chloro-difluoro-methoxy)-phenylamino]-pht...)
Affinity DataIC50: 630nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173051BDBM50173051(4-(4-(3,4-dichlorophenylamino)phthalazin-1-yl)benz...)
Affinity DataIC50: 840nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173024BDBM50173024(4-(4-(4-(chlorodifluoromethoxy)phenylamino)phthala...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173041BDBM50173041(3,5-dimethoxy-N-(1-(naphthalen-2-ylmethyl)piperidi...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173011BDBM50173011(4-(4-(4-chlorophenylamino)phthalazin-1-yl)benzamid...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173029BDBM50173029(4-(4-m-Tolylamino-phthalazin-1-yl)-benzamide | 4-(...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173012BDBM50173012(4-[4-(3-Chloro-phenylamino)-phthalazin-1-yl]-benza...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173017BDBM50173017(4-(4-(p-tolylamino)phthalazin-1-yl)benzamide | 4-(...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173043BDBM50173043(4-[4-(4-Methoxy-phenylamino)-phthalazin-1-yl]-benz...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179886BDBM50179886((4-tert-Butylphenyl)-(4-quinolin-5-yl-phthalazin-1...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173025BDBM50173025(methyl 4-(4-(4-carbamoylphenyl)phthalazin-1-ylamin...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173013BDBM50173013(4-[4-(4-Chloro-phenylamino)-phthalazin-1-yl]-N-met...)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173047BDBM50173047(3-{4-[4-(Chloro-difluoro-methoxy)-phenylamino]-pht...)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173020BDBM50173020((4-{4-[4-(Chloro-difluoro-methoxy)-phenylamino]-ph...)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247683BDBM50247683(4-(4-(4-phenoxyphenylamino)phthalazin-1-yl)benzami...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179895BDBM50179895(4-(isoquinolin-5-yl)-N-o-tolylphthalazin-1-amine |...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173028BDBM50173028(4-[4-(4-Benzyloxy-phenylamino)-phthalazin-1-yl]-be...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173042BDBM50173042(4-[4-(4-carbamoylanilino)-1-phthalazinyl]benzamide...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247684BDBM50247684(4-(4-(4-(N-methylsulfamoyl)phenylamino)phthalazin-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50179887BDBM50179887(N-(4-chlorophenyl)-4-(quinolin-5-yl)phthalazin-1-a...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173016BDBM50173016(4-(4-(phenylamino)phthalazin-1-yl)benzamide | 4-(4...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173050BDBM50173050(4-(4-(4-(trifluoromethoxy)phenylthio)phthalazin-1-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173008BDBM50173008(4-[4-(4-Trifluoromethoxy-phenoxy)-phthalazin-1-yl]...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173037BDBM50173037([4-(Chloro-difluoro-methoxy)-phenyl]-(4-phenyl-pht...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173015BDBM50173015(N-tert-butyl-4-(4-(4-(chlorodifluoromethoxy)phenyl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173009BDBM50173009(4-(4-(4-(chlorodifluoromethoxy)phenylamino)phthala...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173014BDBM50173014([4-(Chloro-difluoro-methoxy)-phenyl]-(4-p-tolyl-ph...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50173018BDBM50173018([4-(Chloro-difluoro-methoxy)-phenyl]-[4-(4-methoxy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Imclone Systems

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247780BDBM50247780(N-(4-(chlorodifluoromethoxy)phenyl)-4-(3-chlorophe...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed