Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50028011
TargetHistone acetyltransferase KAT2B(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50247839(methyl 3-(5-chloro-3-oxoisothiazol-2(3H)-yl)propan...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human recombinant HAT PCAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50247843(Ethyl 3-(5-chloro-3-oxoisothiazol-2(3H)-yl)propano...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human recombinant HAT PCAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50247844(5-Chloro-2-(3-chloro-4-fluorophenyl)isothiazol-3(2...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human recombinant HAT PCAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50247840(Methyl 4-(5-chloro-3-oxoisothiazol-2(3H)-yl)butano...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human recombinant HAT PCAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50247845(Benzyl [2-(5-chloro-3-oxoisothiazol-2(3H)-yl)ethyl...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human recombinant HAT PCAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50247841(Methyl 4-(5-chloro-3-oxoisothiazol-2(3H)-yl)pentan...)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human recombinant HAT PCAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50247838(Methyl 2-(5-chloro-3-oxoisothiazol-2(3H)-yl)ethano...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of human recombinant HAT PCAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50247837(5-Chloro-2-pentylisothiazol-3(2H)-one | CHEMBL4891...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of human recombinant HAT PCAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50247820(5-Chloro-2-ethylisothiazol-3(2H)-one | CHEMBL46147...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant HAT PCAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50247842(Methyl 6-(5-chloro-3-oxoisothiazol-2(3H)-yl)hexano...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of human recombinant HAT PCAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50247868(2-(3-Chloro-4-fluorophenyl)isothiazol-3(2H)-one | ...)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of human recombinant HAT PCAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50247871(Methyl 3-[4-{[(benzyloxy)carbonyl]amino}-5-chloro-...)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of human recombinant HAT PCAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50247869(methyl 3-(5-chloro-1-oxido-3-oxoisothiazol-2(3H)-y...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human recombinant HAT PCAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50247846(2-Ethylisothiazol-3(2H)-one | CHEMBL490685)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant HAT PCAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50247865(Methyl 3-(3-oxoisothiazol-2(3H)-yl)propanoate | CH...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant HAT PCAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50247864(2-pentylisothiazol-3(2H)-one | CHEMBL491668)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant HAT PCAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50247867(methyl 6-(3-oxoisothiazol-2(3H)-yl)hexanoate | CHE...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant HAT PCAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50247866(Methyl 4-(3-oxoisothiazol-2(3H)-yl)butanoate | CHE...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant HAT PCAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50247870(Methyl 3-[(5-chloroisothiazol-3-yl)amino]propanoat...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant HAT PCAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed