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Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 3074
LigandPNGBDBM27641(1-(3-{[(2S)-2-aminopropanamido]methyl}phenyl)-N-[(...)
Affinity DataIC50:  60nMpH: 9.0 T: 22°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM27642(1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-3-y...)
Affinity DataIC50:  60nMpH: 9.0 T: 22°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM27659(1-(3-{[(2S)-2-aminopropanamido]methyl}phenyl)-N-be...)
Affinity DataIC50:  80nMpH: 9.0 T: 22°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM27650(1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-3-y...)
Affinity DataIC50:  220nMpH: 9.0 T: 22°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM27655(1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-2-y...)
Affinity DataIC50:  230nMpH: 9.0 T: 22°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM27651(1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-3-y...)
Affinity DataIC50:  260nMpH: 9.0 T: 22°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM27643(1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-2-y...)
Affinity DataIC50:  300nMpH: 9.0 T: 22°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM27652(1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-3-y...)
Affinity DataIC50:  370nMpH: 9.0 T: 22°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM27653(methyl 2-({[1-(5-{[(2S)-2-aminopropanamido]methyl}...)
Affinity DataIC50:  770nMpH: 9.0 T: 22°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM27649(1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-3-y...)
Affinity DataIC50:  790nMpH: 9.0 T: 22°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM27644(1-(4-{[(2S)-2-aminopropanamido]methyl}-1,3-thiazol...)
Affinity DataIC50:  2.20E+3nMpH: 9.0 T: 22°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM27654(1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-2-y...)
Affinity DataIC50:  2.31E+3nMpH: 9.0 T: 22°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM27657(1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-2-y...)
Affinity DataIC50:  2.92E+3nMpH: 9.0 T: 22°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM27646(1-(6-{[(2S)-2-aminopropanamido]methyl}pyridin-2-yl...)
Affinity DataIC50:  3.05E+3nMpH: 9.0 T: 22°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM27658(1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-3-y...)
Affinity DataIC50:  3.35E+3nMpH: 9.0 T: 22°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM27645(1-(4-{[(2S)-2-aminopropanamido]methyl}pyridin-2-yl...)
Affinity DataIC50:  4.20E+3nMpH: 9.0 T: 22°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM27656(1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-2-y...)
Affinity DataIC50:  4.48E+3nMpH: 9.0 T: 22°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM27647(1-{2-[(2S)-2-aminopropanoyl]-2,3-dihydro-1H-isoind...)
Affinity DataIC50: >1.00E+4nMpH: 9.0 T: 22°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM27648(1-(2-{[(2S)-2-aminopropanamido]methyl}-1-benzofura...)
Affinity DataIC50: >1.00E+4nMpH: 9.0 T: 22°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed