Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50028136
TargetProstaglandin G/H synthase 2(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029613BDBM50029613(1-methoxy-4-[2-(4-methylsulfonylphenyl)-1-cyclopen...)
Affinity DataIC50: 7nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266516BDBM50266516(5-(4-Fluorophenyl)-1-(4-methanesulfonylphenyl)-1H-...)
Affinity DataIC50: 30nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266515BDBM50266515(5-(4-Chlorophenyl)-1-(4-methanesulfonylphenyl)-1H-...)
Affinity DataIC50: 40nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 11639BDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 70nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266511BDBM50266511(1-(4-Methanesulfonylphenyl)-5-phenyl-1H-[1,2,3]tri...)
Affinity DataIC50: 110nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266512BDBM50266512(1-(4-Methanesulfonyl-phenyl)-5-p-tolyl-1H-[1,2,3]t...)
Affinity DataIC50: 120nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266480BDBM50266480(1-(4-Methanesulfonylphenyl)-4-phenyl-1H-[1,2,3]tri...)
Affinity DataIC50: 150nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266513BDBM50266513(5-(4-Methoxyphenyl)-1-(4-(methylsulfonyl)phenyl)-1...)
Affinity DataIC50: 170nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266484BDBM50266484(4-(4-Chlorophenyl)-1-(4-methanesulfonylphenyl)-1H-...)
Affinity DataIC50: 190nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266485BDBM50266485(4-(4-Fluorophenyl)-1-(4-methanesulfonylphenyl)-1H-...)
Affinity DataIC50: 210nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266514BDBM50266514(N,N-dimethyl-4-(1-(4-(methylsulfonyl)phenyl)-1H-[1...)
Affinity DataIC50: 360nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266515BDBM50266515(5-(4-Chlorophenyl)-1-(4-methanesulfonylphenyl)-1H-...)
Affinity DataIC50: 700nMAssay Description:Inhibition of COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266512BDBM50266512(1-(4-Methanesulfonyl-phenyl)-5-p-tolyl-1H-[1,2,3]t...)
Affinity DataIC50: 780nMAssay Description:Inhibition of COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266511BDBM50266511(1-(4-Methanesulfonylphenyl)-5-phenyl-1H-[1,2,3]tri...)
Affinity DataIC50: 810nMAssay Description:Inhibition of COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266513BDBM50266513(5-(4-Methoxyphenyl)-1-(4-(methylsulfonyl)phenyl)-1...)
Affinity DataIC50: 830nMAssay Description:Inhibition of COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266514BDBM50266514(N,N-dimethyl-4-(1-(4-(methylsulfonyl)phenyl)-1H-[1...)
Affinity DataIC50: 840nMAssay Description:Inhibition of COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266516BDBM50266516(5-(4-Fluorophenyl)-1-(4-methanesulfonylphenyl)-1H-...)
Affinity DataIC50: 910nMAssay Description:Inhibition of COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266482BDBM50266482(1-(4-Methanesulfonyl-phenyl)-4-(4-methoxyphenyl)-1...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266481BDBM50266481(1-(4-Methanesulfonyl-phenyl)-4-p-tolyl-1H-[1,2,3]t...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029613BDBM50029613(1-methoxy-4-[2-(4-methylsulfonylphenyl)-1-cyclopen...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 11639BDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266483BDBM50266483({4-[1-(4-Methanesulfonylphenyl)-1H-[1,2,3]triazol-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of COX2 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266482BDBM50266482(1-(4-Methanesulfonyl-phenyl)-4-(4-methoxyphenyl)-1...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266484BDBM50266484(4-(4-Chlorophenyl)-1-(4-methanesulfonylphenyl)-1H-...)
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266485BDBM50266485(4-(4-Fluorophenyl)-1-(4-methanesulfonylphenyl)-1H-...)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266480BDBM50266480(1-(4-Methanesulfonylphenyl)-4-phenyl-1H-[1,2,3]tri...)
Affinity DataIC50: 2.08E+4nMAssay Description:Inhibition of COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266481BDBM50266481(1-(4-Methanesulfonyl-phenyl)-4-p-tolyl-1H-[1,2,3]t...)
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50266483BDBM50266483({4-[1-(4-Methanesulfonylphenyl)-1H-[1,2,3]triazol-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed