Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 4988
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis subsp. mobilis (strain ATCC 3182...)
Philipps-UniversitÄT Marburg

LigandChemical structure of BindingDB Monomer ID 84658BDBM84658(lin-benzoguanine scaffold, 7)
Affinity DataKi:  3.5nMpH: 7.3Assay Description:Inhibition assay using tRNA-guanine transglycosylase (TGT).More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2012
Entry Details Article
PubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis subsp. mobilis (strain ATCC 3182...)
Philipps-UniversitÄT Marburg

LigandChemical structure of BindingDB Monomer ID 84659BDBM84659(lin-benzoguanine scaffold, 8)
Affinity DataKi:  5.5nMpH: 7.3Assay Description:Inhibition assay using tRNA-guanine transglycosylase (TGT).More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2012
Entry Details Article
PubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis subsp. mobilis (strain ATCC 3182...)
Philipps-UniversitÄT Marburg

LigandChemical structure of BindingDB Monomer ID 84657BDBM84657(lin-benzoguanine scaffold, 6)
Affinity DataKi:  5.80nMpH: 7.3Assay Description:Inhibition assay using tRNA-guanine transglycosylase (TGT).More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2012
Entry Details Article
PubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis subsp. mobilis (strain ATCC 3182...)
Philipps-UniversitÄT Marburg

LigandChemical structure of BindingDB Monomer ID 84660BDBM84660(lin-benzoguanine scaffold, 9)
Affinity DataKi:  6nMpH: 7.3Assay Description:Inhibition assay using tRNA-guanine transglycosylase (TGT).More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2012
Entry Details Article
PubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis subsp. mobilis (strain ATCC 3182...)
Philipps-UniversitÄT Marburg

LigandChemical structure of BindingDB Monomer ID 84661BDBM84661(lin-benzoguanine scaffold, 10)
Affinity DataKi:  10nMpH: 7.3Assay Description:Inhibition assay using tRNA-guanine transglycosylase (TGT).More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis subsp. mobilis (strain ATCC 3182...)
Philipps-UniversitÄT Marburg

LigandChemical structure of BindingDB Monomer ID 84656BDBM84656(lin-benzoguanine scaffold, 5)
Affinity DataKi:  77nMpH: 7.3Assay Description:Inhibition assay using tRNA-guanine transglycosylase (TGT).More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2012
Entry Details Article
PubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis subsp. mobilis (strain ATCC 3182...)
Philipps-UniversitÄT Marburg

LigandChemical structure of BindingDB Monomer ID 84655BDBM84655(lin-benzoguanine scaffold, 4)
Affinity DataKi:  1.50E+3nMpH: 7.3Assay Description:Inhibition assay using tRNA-guanine transglycosylase (TGT).More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2012
Entry Details Article
PubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis subsp. mobilis (strain ATCC 3182...)
Philipps-UniversitÄT Marburg

LigandChemical structure of BindingDB Monomer ID 84654BDBM84654(lin-benzoguanine scaffold, 3)
Affinity DataKi:  4.10E+3nMpH: 7.3Assay Description:Inhibition assay using tRNA-guanine transglycosylase (TGT).More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2012
Entry Details Article
PubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis subsp. mobilis (strain ATCC 3182...)
Philipps-UniversitÄT Marburg

LigandChemical structure of BindingDB Monomer ID 84653BDBM84653(Quinazolinone scaffold, 2)
Affinity DataKi:  7.60E+3nMpH: 7.3Assay Description:Inhibition assay using tRNA-guanine transglycosylase (TGT).More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2012
Entry Details Article
PubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis subsp. mobilis (strain ATCC 3182...)
Philipps-UniversitÄT Marburg

LigandChemical structure of BindingDB Monomer ID 84652BDBM84652(Quinazolinone scaffold, 1)
Affinity DataKi:  3.10E+4nMpH: 7.3Assay Description:Inhibition assay using tRNA-guanine transglycosylase (TGT).More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2012
Entry Details Article
PubMed