Compile Data Set for Download or QSAR
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Report error Found 61 Enz. Inhib. hit(s) with all data for entry = 50028286
TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50257829(2-(4-amino-5-(5-iodo-2-isopropyl-4-methoxyphenoxy)...)
Affinity DataIC50:  2nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50257829(2-(4-amino-5-(5-iodo-2-isopropyl-4-methoxyphenoxy)...)
Affinity DataIC50:  5nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413367(CHEMBL523173)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413347(CHEMBL494353)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413346(CHEMBL494160)
Affinity DataIC50:  7.90nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50257636(5-(5-iodo-2-isopropyl-4-methoxyphenoxy)pyrimidine-...)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413367(CHEMBL523173)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50257636(5-(5-iodo-2-isopropyl-4-methoxyphenoxy)pyrimidine-...)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413364(CHEMBL492300)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413356(CHEMBL492933)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413349(CHEMBL494582)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413345(CHEMBL494159)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413364(CHEMBL492300)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413357(CHEMBL492934)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413367(CHEMBL523173)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413366(CHEMBL492907)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413345(CHEMBL494159)
Affinity DataIC50:  25nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413346(CHEMBL494160)
Affinity DataIC50:  32nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413367(CHEMBL523173)
Affinity DataIC50:  32nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413347(CHEMBL494353)
Affinity DataIC50:  32nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50257636(5-(5-iodo-2-isopropyl-4-methoxyphenoxy)pyrimidine-...)
Affinity DataIC50:  39.8nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50257636(5-(5-iodo-2-isopropyl-4-methoxyphenoxy)pyrimidine-...)
Affinity DataIC50:  39.8nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413356(CHEMBL492933)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413357(CHEMBL492934)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413352(CHEMBL443930)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413349(CHEMBL494582)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413365(CHEMBL492703)
Affinity DataIC50:  63nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413365(CHEMBL492703)
Affinity DataIC50:  63nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413360(CHEMBL492745)
Affinity DataIC50:  63nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413366(CHEMBL492907)
Affinity DataIC50:  63nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413353(CHEMBL493741)
Affinity DataIC50:  79nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413363(CHEMBL492299)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413348(CHEMBL494581)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413362(CHEMBL493547)
Affinity DataIC50:  126nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413358(CHEMBL492935)
Affinity DataIC50:  158nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413361(CHEMBL493546)
Affinity DataIC50:  158nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413353(CHEMBL493741)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413352(CHEMBL443930)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413360(CHEMBL492745)
Affinity DataIC50:  251nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413358(CHEMBL492935)
Affinity DataIC50:  251nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413355(CHEMBL492729)
Affinity DataIC50:  251nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413368(CHEMBL523000)
Affinity DataIC50:  251nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413363(CHEMBL492299)
Affinity DataIC50:  316nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413350(CHEMBL492789)
Affinity DataIC50:  398nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413361(CHEMBL493546)
Affinity DataIC50:  398nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413359(CHEMBL492744)
Affinity DataIC50:  398nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413362(CHEMBL493547)
Affinity DataIC50:  398nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413368(CHEMBL523000)
Affinity DataIC50:  631nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413348(CHEMBL494581)
Affinity DataIC50:  794nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Human)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413359(CHEMBL492744)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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