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Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50028314
TargetNeurotensin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50276349(CHEMBL450740 | Polyamine-NT)
Affinity DataKi:  2.50E+5nMAssay Description:Binding affinity to human recombinant NTS1 in HEK293T cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeurotensin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50276349(CHEMBL450740 | Polyamine-NT)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human recombinant NTS1 receptor expressed in HEK293 cells assessed as stimulation of Ca2+ mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeurotensin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50276350(((N-methyl-Arg)-Lys-Pro-(L-neo-Trp)-(tert-Leu)-Leu...)
Affinity DataKd:  1.55nMAssay Description:Binding affinity to human recombinant NTS1 in HEK293T cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeurotensin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50241512(CHEMBL270332 | c(Lys-Lys-Pro-Tyr-Ile-Leu-Lys-Lys-P...)
Affinity DataKd:  150nMAssay Description:Binding affinity to human recombinant NTS1 in HEK293T cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed