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Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50028337
TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276150(2-(2,2,6,6-Tetramethyl-1,2,3,6-tetrahydropyridin-4...)
Affinity DataIC50:  14nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276874(2-(1-Oxyl-2,2,6,6-tetramethyl-1,2,3,6-tetrahydropy...)
Affinity DataIC50:  26nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276945(2-(1,2,2,5,5-pentamethyl-2,5-dihydro-1H-pyrrol-3-y...)
Affinity DataIC50:  42nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276946(2-(1-Acetyl-2,2,5,5-pentamethyl-2,5-dihydro-1H-pyr...)
Affinity DataIC50:  49nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276947(2-(1-Methoxy-2,2,5,5-pentamethyl-2,5-dihydro-1H-py...)
Affinity DataIC50:  61nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276872(2-[4-(1-Oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-py...)
Affinity DataIC50:  78nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276148(2-[4-(2,2,5,5-Tetramethyl-2,5-dihydro-1H-pyrrol-3-...)
Affinity DataIC50:  98nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276112(2-[4-(3-Trifluoromethylphenyl)-2,2,5,5-tetramethyl...)
Affinity DataIC50:  133nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276110(2-(4-Bromo-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrr...)
Affinity DataIC50:  137nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276201(2-[1-Oxyl-4-(3-trifluoromethylphenyl)-2,2,5,5-tetr...)
Affinity DataIC50:  149nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276199(2-(4-Bromo-1-oxyl-2,2,5,5-tetramethyl-2,5-dihydro-...)
Affinity DataIC50:  201nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276109(4-(4-Carbamoyl-1H-benzimidazol-2-yl)-2,2,5,5-tetra...)
Affinity DataIC50:  216nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276111(2-(4-Phenyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyr...)
Affinity DataIC50:  310nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276108(2-(2,2,5,5-Tetramethyl-2,5-dihydro-1H-pyrrol-3-yl)...)
Affinity DataIC50:  345nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276203(2-(4,4,6,6-Tetramethyl-5,6-dihydro-4H-thieno[3,4-c...)
Affinity DataIC50:  354nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276202(2-[4-(2,2,5,5-Tetramethyl-2,5-dihydro-1H-pyrrol-3-...)
Affinity DataIC50:  432nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276204(2-(1,1,3,3-Tetramethyl-2,3-dihydro-1H-isoindol-5-y...)
Affinity DataIC50:  450nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276205(2-(1,1,3,3-Tetramethyl-2,3-dihydro-1H-pyrrolo[3,4-...)
Affinity DataIC50:  470nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276943(2-[4-(1-Oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-py...)
Affinity DataIC50:  472nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276875(2-[4-(1-Oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-py...)
Affinity DataIC50:  564nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276151(2-[4-(2,2,5,5-Tetramethyl-2,5-dihydro-1H-pyrrol-3-...)
Affinity DataIC50:  572nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276197(2-(1-Oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrro...)
Affinity DataIC50:  721nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276200(2-(1-Oxyl-4-phenyl-2,2,5,5-tetramethyl-2,5-dihydro...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276873(2-[4-Dibenzofuran-4-yl-1-oxyl-2,2,5,5-tetramethyl-...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276149(2-[4-Dibenzofuran-4-yl-2,2,5,5-tetramethyl-2,5-dih...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276114(2-((2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrrol-3-yl...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276944(2-(5-Oxyl-4,4,6,6-tetramethyl-5,6-dihydro-4H-thien...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276113(2-((2,2,6,6-tetramethyl-1,2,3,6-tetrahydropyridin-...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50413274(CHEMBL2094004)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50413275(CHEMBL2094005)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276116(2-(1-Oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrro...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276115(1-(1-Oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrro...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPoly [ADP-ribose] polymerase 1(Rat)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276152(2-(2,2,5,5-Tetramethyl-2,5-dihydro-1H-pyrrol-3-yl)...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed