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Report error Found 62 Enz. Inhib. hit(s) with all data for entry = 50041699
TargetBeta-2 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human cloned beta2 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
PDB3D3D Structure (crystal)

TargetBeta-1 adrenergic receptor(Guinea pig)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413483(CHEMBL514032)
Affinity DataEC50:  10nMAssay Description:Agonist activity at beta-1 adrenergic receptor in guinea pig trachea assessed as inhibition of electrical stimulation-induced muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413487(CHEMBL516056)
Affinity DataEC50:  794nMAssay Description:Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413488(CHEMBL474393)
Affinity DataEC50:  631nMAssay Description:Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413489(CHEMBL500782)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413491(CHEMBL456485)
Affinity DataEC50:  631nMAssay Description:Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413490(CHEMBL506518)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM25771(1-hydroxy-2-naphthoic acid;4-[1-hydroxy-2-[6-(4-ph...)
Affinity DataEC50:  0.251nMAssay Description:Agonist activity at human cloned beta2 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
PDB3D3D Structure (crystal)

TargetBeta-1 adrenergic receptor(Guinea pig)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413484(CHEMBL475389)
Affinity DataEC50:  2nMAssay Description:Agonist activity at beta-1 adrenergic receptor in guinea pig trachea assessed as inhibition of electrical stimulation-induced muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413485(CHEMBL446840 | CHEMBL483200)
Affinity DataEC50:  316nMAssay Description:Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413480(CHEMBL520313)
Affinity DataEC50:  251nMAssay Description:Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413482(CHEMBL443435)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413496(CHEMBL483407)
Affinity DataEC50:  7.94E+4nMAssay Description:Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM25771(1-hydroxy-2-naphthoic acid;4-[1-hydroxy-2-[6-(4-ph...)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413482(CHEMBL443435)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413485(CHEMBL446840 | CHEMBL483200)
Affinity DataEC50:  1.59E+3nMAssay Description:Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413483(CHEMBL514032)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413496(CHEMBL483407)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413480(CHEMBL520313)
Affinity DataEC50:  501nMAssay Description:Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM86453(CAS_73573-87-2 | Formoterol | NSC_3083544)
Affinity DataEC50:  0.501nMAssay Description:Agonist activity at human cloned beta2 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank


TargetBeta-2 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413493(CHEMBL475237)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human cloned beta2 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413483(CHEMBL514032)
Affinity DataEC50:  0.501nMAssay Description:Agonist activity at human cloned beta2 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413481(CHEMBL474616 | CHEMBL485847)
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at human cloned beta2 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Guinea pig)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413485(CHEMBL446840 | CHEMBL483200)
Affinity DataEC50:  0.794nMAssay Description:Agonist activity at beta-1 adrenergic receptor in guinea pig trachea assessed as inhibition of electrical stimulation-induced muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413495(CHEMBL483202)
Affinity DataEC50:  7.90nMAssay Description:Agonist activity at human cloned beta2 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413492(CHEMBL475236)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human cloned beta2 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Guinea pig)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413480(CHEMBL520313)
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at beta-1 adrenergic receptor in guinea pig trachea assessed as inhibition of electrical stimulation-induced muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413495(CHEMBL483202)
Affinity DataEC50:  2.51E+3nMAssay Description:Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413492(CHEMBL475236)
Affinity DataEC50:  5.01E+3nMAssay Description:Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413492(CHEMBL475236)
Affinity DataEC50:  2.00E+4nMAssay Description:Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413493(CHEMBL475237)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413481(CHEMBL474616 | CHEMBL485847)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413481(CHEMBL474616 | CHEMBL485847)
Affinity DataEC50:  316nMAssay Description:Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413495(CHEMBL483202)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413493(CHEMBL475237)
Affinity DataEC50:  2.51E+3nMAssay Description:Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413482(CHEMBL443435)
Affinity DataEC50:  0.158nMAssay Description:Agonist activity at human cloned beta2 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413480(CHEMBL520313)
Affinity DataEC50:  0.794nMAssay Description:Agonist activity at human cloned beta2 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
PDB3D3D Structure (crystal)

TargetBeta-3 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM86453(CAS_73573-87-2 | Formoterol | NSC_3083544)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Guinea pig)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM25771(1-hydroxy-2-naphthoic acid;4-[1-hydroxy-2-[6-(4-ph...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at beta-1 adrenergic receptor in guinea pig trachea assessed as inhibition of electrical stimulation-induced muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Guinea pig)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413481(CHEMBL474616 | CHEMBL485847)
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at beta-1 adrenergic receptor in guinea pig trachea assessed as inhibition of electrical stimulation-induced muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413496(CHEMBL483407)
Affinity DataEC50:  2.51E+4nMAssay Description:Agonist activity at human cloned beta2 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM86453(CAS_73573-87-2 | Formoterol | NSC_3083544)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Guinea pig)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413482(CHEMBL443435)
Affinity DataEC50:  0.0398nMAssay Description:Agonist activity at beta-1 adrenergic receptor in guinea pig trachea assessed as inhibition of electrical stimulation-induced muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413485(CHEMBL446840 | CHEMBL483200)
Affinity DataEC50:  0.158nMAssay Description:Agonist activity at human cloned beta2 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413483(CHEMBL514032)
Affinity DataEC50:  316nMAssay Description:Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)
Affinity DataEC50:  7.90nMAssay Description:Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank


TargetBeta-1 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM25771(1-hydroxy-2-naphthoic acid;4-[1-hydroxy-2-[6-(4-ph...)
Affinity DataEC50:  794nMAssay Description:Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413489(CHEMBL500782)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-1 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413490(CHEMBL506518)
Affinity DataEC50:  126nMAssay Description:Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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