Compile Data Set for Download or QSAR
maximum 50k data
Found 24 Enz. Inhib. hit(s) with all data for entry = 50028590
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50276347((+/-)-1,1,1-trifluoro-3-(2-(3-(1,1,2,2-tetrafluoro...)
Affinity DataIC50:  33nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50276347((+/-)-1,1,1-trifluoro-3-(2-(3-(1,1,2,2-tetrafluoro...)
Affinity DataIC50:  33nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50277885(CHEMBL490868 | Tetrahydroquinline A)
Affinity DataIC50:  39nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50277959(3-(5-(3-chlorophenyl)-2-(3-(1,1,2,2-te trafluoroet...)
Affinity DataIC50:  64nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50278012(1,1,1-tri fluoro-3-(2-(3-(1,1,2,2-tetrafluoroethox...)
Affinity DataIC50:  96nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50278011(1,1,1-trifluoro-3-(5-(3-fluorophenyl) -2-(3-(1,1,2...)
Affinity DataIC50:  117nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50277884((R)-1-((R)-2,5-bis(3-(trifluoromethoxy)phenyl)-3,4...)
Affinity DataIC50:  125nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50277727(3-(2,5-bis(3-(trifluoromethoxy) phenyl)-3,4-dihydr...)
Affinity DataIC50:  125nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50278055(1,1,1-trifluoro -3-(5-(3-methoxyphenyl)-2-(3-(1,1,...)
Affinity DataIC50:  126nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50277688(1,1,1-trifluoro-3-(5-(3-(trifluoromethoxy)phenyl)-...)
Affinity DataIC50:  143nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50277688(1,1,1-trifluoro-3-(5-(3-(trifluoromethoxy)phenyl)-...)
Affinity DataIC50:  143nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50277459(3-(2-(3-(1,1,2,2-tetrafluoroethoxy)phenyl )-1-(3,3...)
Affinity DataIC50:  235nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50277812(1-(2,5-bis(3-(trifluoromethoxy) phenyl)-3,4-dihydr...)
Affinity DataIC50:  326nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50277773(1-(2,5-bis(3-(trifluoromethoxy)phenyl)-3,4-dihydro...)
Affinity DataIC50:  331nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50277921(3-(5-(2,3-dichlorophenyl )-2-(3-(1,1,2,2-tetrafluo...)
Affinity DataIC50:  400nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50277460(1,1,1-trifluoro-3-(2-(3-(1,1,2,2-tetrafluoroethoxy...)
Affinity DataIC50:  500nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50276280(3-(5-(4-chloro-3-ethylphenoxy)-2 -(3-(1,1,2,2-tetr...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50276280(3-(5-(4-chloro-3-ethylphenoxy)-2 -(3-(1,1,2,2-tetr...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50277811(1-(2,5-bis(3-(trifluoromethoxy)phenyl)-3,4-dihydro...)
Affinity DataIC50:  744nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50277492(1,1,1-trifluoro-3-(5-(pyridin-3-yl)-2-(3-(1,1,2,2-...)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50277886(CHEMBL491072 | Tetrahydroquinoline B)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50277557(1,1,1-trifluoro-3-(5-(3-isopropylphenyl)-2-(3-(1,1...)
Affinity DataIC50:  2.77E+5nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50277556(1,1,1-trifluoro-3-(2-(3-(1,1,2,2-tetrafluoroethoxy...)
Affinity DataIC50:  3.17E+5nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50277558(1,1,1-trifluoro-3-(5-(3-isopropoxyphenyl)-2-(3-(1,...)
Affinity DataIC50:  3.45E+5nMAssay Description:Inhibition of human plasma derived CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed