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Found 10 Enz. Inhib. hit(s) with all data for entry = 50028604
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277598(CHEMBL453211 | N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)p...)
Affinity DataIC50:  9nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277599(CHEMBL507541 | N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)p...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277597(CHEMBL501242 | N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)p...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277595(CHEMBL445281 | N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)p...)
Affinity DataIC50:  15nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277594(CHEMBL448015 | N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)p...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277596(CHEMBL504917 | N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)p...)
Affinity DataIC50:  24nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50234644(CHEMBL400043 | N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)p...)
Affinity DataIC50:  50nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50234646(2-(((2S,3S)-4-(3-(2H-tetrazol-5-yl)phenylamino)-3-...)
Affinity DataIC50:  96nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50234643(CHEMBL399839 | N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)p...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50234645(CHEMBL253865 | N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)p...)
Affinity DataIC50:  360nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed