Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 3215
LigandPNGBDBM29407(7-alkoxyisoquinoline, 17)
Affinity DataIC50:  100nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29411(7-alkoxyisoquinoline, 21)
Affinity DataIC50:  100nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29410(7-alkoxyisoquinoline, 20)
Affinity DataIC50:  126nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29421(7-alkoxyisoquinoline, 31)
Affinity DataIC50:  158nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29423(7-alkoxyisoquinoline, 33)
Affinity DataIC50:  158nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29408(7-alkoxyisoquinoline, 18)
Affinity DataIC50:  398nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

LigandPNGBDBM29412(7-alkoxyisoquinoline, 22)
Affinity DataIC50:  398nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29420(7-alkoxyisoquinoline, 30)
Affinity DataIC50:  631nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29425(7-alkoxyisoquinoline, 35)
Affinity DataIC50:  631nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29409(7-alkoxyisoquinoline, 19)
Affinity DataIC50:  794nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29422(7-alkoxyisoquinoline, 32)
Affinity DataIC50:  794nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29418(7-alkoxyisoquinoline, 28)
Affinity DataIC50:  1.00E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29416(7-alkoxyisoquinoline, 26)
Affinity DataIC50:  1.26E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29406(7-alkoxyisoquinoline, 16)
Affinity DataIC50:  1.26E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29424(7-alkoxyisoquinoline, 34)
Affinity DataIC50:  1.26E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29426(7-alkoxyisoquinoline, 36)
Affinity DataIC50:  1.26E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29417(7-alkoxyisoquinoline, 27)
Affinity DataIC50:  2.00E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29427(7-alkoxyisoquinoline, 37)
Affinity DataIC50:  2.51E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29411(7-alkoxyisoquinoline, 21)
Affinity DataIC50:  2.51E+3nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29421(7-alkoxyisoquinoline, 31)
Affinity DataIC50:  3.16E+3nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29431(benzyloxyisoquinoline, 7)
Affinity DataIC50:  3.16E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29415(7-alkoxyisoquinoline, 25)
Affinity DataIC50:  3.16E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29408(7-alkoxyisoquinoline, 18)
Affinity DataIC50:  3.98E+3nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

LigandPNGBDBM29420(7-alkoxyisoquinoline, 30)
Affinity DataIC50:  3.98E+3nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29428(7-alkoxyisoquinoline, 38)
Affinity DataIC50:  3.98E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

LigandPNGBDBM29413(7-alkoxyisoquinoline, 23)
Affinity DataIC50:  5.01E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

LigandPNGBDBM29429(7-alkoxyisoquinoline, 39)
Affinity DataIC50:  5.01E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

LigandPNGBDBM29423(7-alkoxyisoquinoline, 33)
Affinity DataIC50:  5.01E+3nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29419(7-alkoxyisoquinoline, 29)
Affinity DataIC50:  5.01E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

LigandPNGBDBM29410(7-alkoxyisoquinoline, 20)
Affinity DataIC50:  6.31E+3nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29406(7-alkoxyisoquinoline, 16)
Affinity DataIC50:  7.94E+3nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29407(7-alkoxyisoquinoline, 17)
Affinity DataIC50:  7.94E+3nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29430(benzyloxyisoquinoline, 6)
Affinity DataIC50:  7.94E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29412(7-alkoxyisoquinoline, 22)
Affinity DataIC50:  1.00E+4nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29424(7-alkoxyisoquinoline, 34)
Affinity DataIC50:  1.00E+4nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29426(7-alkoxyisoquinoline, 36)
Affinity DataIC50:  1.00E+4nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29417(7-alkoxyisoquinoline, 27)
Affinity DataIC50:  1.26E+4nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29409(7-alkoxyisoquinoline, 19)
Affinity DataIC50:  1.26E+4nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29414(7-alkoxyisoquinoline, 24)
Affinity DataIC50:  1.26E+4nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29422(7-alkoxyisoquinoline, 32)
Affinity DataIC50:  1.26E+4nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29415(7-alkoxyisoquinoline, 25)
Affinity DataIC50:  1.58E+4nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29425(7-alkoxyisoquinoline, 35)
Affinity DataIC50:  1.58E+4nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29427(7-alkoxyisoquinoline, 37)
Affinity DataIC50:  2.00E+4nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29430(benzyloxyisoquinoline, 6)
Affinity DataIC50: >2.51E+4nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29413(7-alkoxyisoquinoline, 23)
Affinity DataIC50: >2.51E+4nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

LigandPNGBDBM29414(7-alkoxyisoquinoline, 24)
Affinity DataIC50: >2.51E+4nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29416(7-alkoxyisoquinoline, 26)
Affinity DataIC50: >2.51E+4nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29431(benzyloxyisoquinoline, 7)
Affinity DataIC50: >2.51E+4nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM29419(7-alkoxyisoquinoline, 29)
Affinity DataIC50: >2.51E+4nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

LigandPNGBDBM29428(7-alkoxyisoquinoline, 38)
Affinity DataIC50: >2.51E+4nMpH: 7.4 T: 22°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

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