Compile Data Set for Download or QSAR
Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 50028697
TargetAdenosine receptor A1(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258734BDBM50258734([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258672BDBM50258672([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258762BDBM50258762([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258734BDBM50258734([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258707BDBM50258707([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258620BDBM50258620([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258620BDBM50258620([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258675BDBM50258675([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258763BDBM50258763([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258709BDBM50258709([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258737BDBM50258737([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258621BDBM50258621([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  9.5nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258672BDBM50258672([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258673BDBM50258673([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258763BDBM50258763([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258672BDBM50258672([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  10.5nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258706BDBM50258706([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  11.5nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258806BDBM50258806([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1-methyl-3-propyl...)
Affinity DataKi:  13.8nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258673BDBM50258673([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  15.1nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258708BDBM50258708([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  16.2nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258621BDBM50258621([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  17.8nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258675BDBM50258675([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  18.2nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258709BDBM50258709([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  20.4nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258762BDBM50258762([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  21.9nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258765BDBM50258765([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258765BDBM50258765([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  28.2nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258709BDBM50258709([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  28.8nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258620BDBM50258620([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  34.7nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258737BDBM50258737([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  35.5nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258805BDBM50258805([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  42.7nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258707BDBM50258707([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  43.7nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258805BDBM50258805([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  50.1nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258734BDBM50258734([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  71nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258621BDBM50258621([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  72.4nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258674BDBM50258674([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  81.3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258734BDBM50258734([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  118nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258706BDBM50258706([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258620BDBM50258620([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  275nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258709BDBM50258709([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  331nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258672BDBM50258672([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  363nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258764BDBM50258764([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  447nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258674BDBM50258674([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  490nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258735BDBM50258735([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  501nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258736BDBM50258736([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  602nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258621BDBM50258621([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  871nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258708BDBM50258708([4-(2,3,4,5-Tetrahydro-1,3-dimethyl-2,4-dioxo-1H-p...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258736BDBM50258736([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  2.24E+3nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universidade De Santiago De Compostela

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258735BDBM50258735([4-(2,3,4,5-Tetrahydro-2,4-dioxo-1,3-dipropyl-1H-p...)
Affinity DataKi:  3.31E+3nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HeLa cells by beta scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed